SCHEMBL2565015

SCHEMBL2565015

c1cc2c(cn1)CCNC2

nearest known ligand 0.77

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.77
CHRNA4 P43681 1/20 0.77
PNMT P11086 6/20 0.54
SIGMAR1 Q99720 1/20 0.54
CD44 P16070 1/20 0.54
MAOB P27338 1/20 0.54
ASIC3 Q9UHC3 3/20 0.46
PKN2 Q16513 1/20 0.45
DRD2 P14416 2/20 0.43
DRD3 P35462 2/20 0.43
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30183351 1.00 CHRNB2 (0.77) CHRNB2CHRNA4PNMTSIGMAR1CD44
Hydrochloric Acid SCHEMBL29759853 0.98 CHRNB2 (0.74) CHRNB2CHRNA4PNMTSIGMAR1CD44
Hydrochloric Acid SCHEMBL785959 0.98 CHRNB2 (0.74) CHRNB2CHRNA4PNMTSIGMAR1CD44
SCHEMBL29850369 0.92 CHRNB2 (0.77) CHRNB2CHRNA4PNMTSIGMAR1CD44
SCHEMBL587887 0.92 CHRNB2 (0.77) CHRNB2CHRNA4PNMTSIGMAR1CD44
Hydrochloric Acid SCHEMBL15238605 0.90 CHRNB2 (0.74) CHRNB2CHRNA4PNMTSIGMAR1CD44
Hydrochloric Acid SCHEMBL4790441 0.90 CHRNB2 (0.74) CHRNB2CHRNA4PNMTSIGMAR1CD44
SCHEMBL19194503 0.88 SIGMAR1 (0.61) CHRNB2CHRNA4PNMTSIGMAR1CD44
SCHEMBL19200207 0.87 CHRNB2 (1.00) CHRNB2CHRNA4PNMTSIGMAR1CD44
SCHEMBL1118591 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 524 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111655695-B Substituted furopyrimidine compounds as PDE1 inhibitors 达特神经科学有限公司 2025-05-27 CN claimed
EP-3717488-A1 SUBSTITUTED FURANOPYRIMIDINE COMPOUNDS AS PDE1 INHIBITORS Dart NeuroScience, LLC (US) 2020-10-07 EP claimed
CN-111655695-A Substituted furopyrimidines as PDE1 inhibitors 达特神经科学有限公司 2020-09-11 CN claimed
EP-3129371-B1 INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 (CDK7) SYROS PHARMACEUTICALS INC (US) 2020-07-29 EP claimed
WO-2019104285-A1 SUBSTITUTED FURANOPYRIMIDINE COMPOUNDS AS PDE1 INHIBITORS DART NEUROSCIENCE, LLC (US) 2019-05-31 WO claimed
US-20100130495-A1 COMPOUNDS 563 ASTRAZENECA AB (SE) 2010-05-27 US claimed
EP-1899334-A2 NAPHTHYRIDINE COMPOUNDS JANSSEN PHARMACEUTICA N.V. (BE) 2008-03-19 EP claimed
WO-2006138714-A2 NAPHTHYRIDINE COMPOUNDS JANSSEN PHARMACEUTICA N.V. (BE) 2006-12-28 WO claimed
US-12629358-B2 Compound used as RET kinase inhibitor and application thereof TYK MEDICINES, INC. (CN) 2026-05-19 US disclosed
US-12624043-B2 Compositions useful for treating disorders related to kit BLUEPRINT MEDICINES CORPORATION (US) 2026-05-12 US disclosed
EP-4155304-B9 COMPOUND USED AS RET KINASE INHIBITOR AND APPLICATION THEREOF TYK MEDICINES INC (CN) 2026-04-15 EP disclosed
US-12595265-B2 Inhibitors of activin receptor-like kinase BLUEPRINT MEDICINES CORPORATION (US) 2026-04-07 US disclosed
EP-4714948-A1 COMPOUND USED FOR EGFR PROTEIN DEGRADATION, AND USE THEREOF TYK Medicines, Inc. (CN) 2026-03-25 EP disclosed
US-12583856-B2 Inhibitors of protein kinase A BLUEPRINT MEDICINES CORPORATION (US) 2026-03-24 US disclosed
WO-2001044250-A1 SUBSTITUTED 1,2,3-TRIAZOLO[1,5-a]QUINAZOLINES FOR ENHANCING COGNITION MERCK SHARP & DOHME LIMITED (GB) 2001-06-21 WO disclosed
EP-0321191-B1 Heterocyclic-substituted quinoline-carboxylic acids PFIZER (US) 1994-11-02 EP disclosed
US-5214051-A Thiazolyl and oxazolyl[5,4-c]piperidyl-substituted quinolone-carboxylic acid and related analogs thereof having antibacterial properties are disclosed PFIZER INC. (US) 1993-05-25 US disclosed
US-5037834-A Heterocycylic-substituted quinoline-carboxylic acids PFIZER INC. (US) 1991-08-06 US disclosed
WO-1989005643-A1 HETEROCYCLIC-SUBSTITUTED QUINOLINE-CARBOXYLIC ACIDS PFIZER INC. (US) 1989-06-29 WO disclosed
EP-0321191-A2 Heterocyclic-substituted quinoline-carboxylic acids PFIZER INC. (US) 1989-06-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12624043-B2 Compositions useful for treating disorders related to kit KIT, RET, SLC26A4 CHRNB2 1417/4885CHRNA4 1339/4885PNMT 1096/4885
US-12583856-B2 Inhibitors of protein kinase A CSNK1A1, CSNK1A1L, CSNK1G1 CHRNB2 1646/4885CHRNA4 1385/4885PNMT 4642/4885
US-20100130495-A1 COMPOUNDS 563 BACE1, PSEN1, PSEN2 CHRNB2 43/4885CHRNA4 85/4885PNMT 270/4885
US-12595265-B2 Inhibitors of activin receptor-like kinase ACVR1, ACVRL1, ACVR2A CHRNB2 89/4885CHRNA4 403/4885PNMT 4593/4885
US-12629358-B2 Compound used as RET kinase inhibitor and application thereof RET, ALK, FGFR3 CHRNB2 1839/4885CHRNA4 2237/4885PNMT 4558/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.