SCHEMBL256579

SCHEMBL256579

COc1cc2[nH]cc(N)c(=O)c2cc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.50
MAPK1 P28482 1/20 0.50
PDPK1 O15530 1/20 0.46
POLB P06746 1/20 0.46
ALDH1A1 P00352 4/20 0.45
HPGD P15428 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
MAPT P10636 3/20 0.44
LMNA P02545 1/20 0.44
GRIN2D O15399 1/20 0.44
GRIN3B O60391 1/20 0.44
GRIN1 Q05586 1/20 0.44
GRIN2A Q12879 1/20 0.44
GRIN2B Q13224 1/20 0.44
GRIN2C Q14957 1/20 0.44
GRIN3A Q8TCU5 1/20 0.44
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
MPO P05164 1/20 0.42
XDH P47989 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL256578 0.83 CTSL (0.64) PDPK1POLBALDH1A1HPGDSMN1; SMN2
SCHEMBL19147143 0.81 KDM4E (0.51) KDM4EMAPK1PDPK1POLBALDH1A1
SCHEMBL6786495 0.79 KDM4E (0.50) KDM4EMAPK1PDPK1POLBALDH1A1
SCHEMBL2749368 0.79 KDM4E (0.50) KDM4EMAPK1PDPK1POLBALDH1A1
SCHEMBL6783400 0.79 KDM4E (0.50) KDM4EMAPK1PDPK1POLBALDH1A1
SCHEMBL7282665 0.76 MTNR1A (0.53) KDM4EMAPK1POLBALDH1A1HPGD
SCHEMBL4765036 0.76 KDM4E (0.47) KDM4EMAPK1PDPK1POLBALDH1A1
SCHEMBL9424983 0.76 KDM4E (0.64) KDM4EMAPK1POLBALDH1A1HPGD
SCHEMBL6434901 0.74 KDM4E (0.48) KDM4EMAPK1PDPK1POLBALDH1A1
SCHEMBL2736689 0.74 PDPK1 (0.41) KDM4EPDPK1ALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012028233-A1 IMIDAZO[4,5-C]QUINOLINES AS DNA-PK INHIBITORS MERCK PATENT GMBH (DE) 2012-03-08 WO disclosed