SCHEMBL2736689

SCHEMBL2736689

COc1cc2c(N)c[nH]c2cc1C

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.41
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
ATM Q13315 1/20 0.39
HTR2A P28223 2/20 0.38
HTR1A P08908 2/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
EGFR P00533 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16473797 0.83 KDM4E (0.42) PDPK1KDM4EMAPTATMHTR1A
SCHEMBL2737054 0.81 HTR1A (0.55) HTR2AHTR1AHTR2CHTR2BEGFR
SCHEMBL188260 0.75 SRC (0.43) KDM4EMAPTATMALDH1A1
SCHEMBL17417809 0.75 PRKAG1 (0.53) KDM4EALDH1A1
SCHEMBL9732348 0.75 ALDH1A1 (0.56) PDPK1KDM4EMAPTALDH1A1
SCHEMBL2736978 0.75 IMPDH2 (0.45) KDM4EMAPTHTR2AALDH1A1MEN1
SCHEMBL23207583 0.74 IDO1 (0.46) ATMHTR2AHTR2CEGFRMEN1
SCHEMBL256579 0.74 KDM4E (0.50) PDPK1KDM4EMAPTALDH1A1MEN1
SCHEMBL31077721 0.73 PRKAB2 (0.43) KDM4E
SCHEMBL4419308 0.73 IMPDH2 (0.34) KDM4EMAPTHTR2AHTR2CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402314-A1 (Aza)indole derivative and use thereof for medical purposes Kissei Pharmaceutical Co., Ltd. (JP) 2012-01-04 EP disclosed