SCHEMBL256578

SCHEMBL256578

COc1cc2[nH]cc(N)c(=O)c2cc1OCc1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 3/20 0.64
CTSV O60911 2/20 0.64
POLB P06746 1/20 0.54
HPGD P15428 3/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
ALDH1A1 P00352 2/20 0.52
LMNA P02545 1/20 0.52
MAPT P10636 1/20 0.52
SRD5A1 P18405 1/20 0.49
SRD5A2 P31213 1/20 0.49
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
MDH2 P40926 1/20 0.44
ELANE P08246 1/20 0.44
SMPD1 P17405 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
IRAK1 P51617 1/20 0.43
IRAK4 Q9NWZ3 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2063876 0.86 CTSV (0.64) CTSLCTSVPOLBHPGDSMN1; SMN2
SCHEMBL256579 0.83 KDM4E (0.50) CTSLCTSVPOLBHPGDSMN1; SMN2
SCHEMBL5458919 0.83 CTSL (0.60) CTSLCTSVPOLBHPGDSMN1; SMN2
SCHEMBL2063188 0.83 CTSV (0.60) CTSLCTSVPOLBHPGDSMN1; SMN2
SCHEMBL248836 0.82 CTSV (0.59) CTSLCTSVPOLBHPGDSMN1; SMN2
SCHEMBL17067000 0.81 CTSV (0.58) CTSLCTSVPOLBHPGDSMN1; SMN2
SCHEMBL18474478 0.81 CTSV (0.57) CTSLCTSVPOLBHPGDSMN1; SMN2
SCHEMBL15730198 0.81 CTSV (0.57) CTSLCTSVPOLBHPGDSMN1; SMN2
SCHEMBL18975225 0.81 SRD5A1 (0.60) CTSLCTSVPOLBHPGDSMN1; SMN2
SCHEMBL187798 0.80 CTSV (0.56) CTSLCTSVPOLBHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012028233-A1 IMIDAZO[4,5-C]QUINOLINES AS DNA-PK INHIBITORS MERCK PATENT GMBH (DE) 2012-03-08 WO disclosed