SCHEMBL256609

SCHEMBL256609

C=C(O)c1cc(F)cnc1Cl

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
AGBL2 Q5U5Z8 1/20 0.33
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
HCAR2 Q8TDS4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL256606 0.82 SCN5A (0.31) SCN5ASCN9A
SCHEMBL27598069 0.80 KEAP1 (0.53) SCN5ASCN9AAGBL2KEAP1NFE2L2
SCHEMBL290570 0.80 KEAP1 (0.53) SCN5ASCN9AAGBL2KEAP1NFE2L2
SCHEMBL31349524 0.80 KEAP1 (0.53) SCN5ASCN9AAGBL2KEAP1NFE2L2
SCHEMBL8357219 0.76 SCN5A (0.36) SCN5ASCN9AAGBL2KEAP1NFE2L2
SCHEMBL4966985 0.76 ALDH1A1 (0.36) SCN5ASCN9AAGBL2KEAP1NFE2L2
SCHEMBL9928617 0.74 AGBL2 (0.39) SCN5ASCN9AAGBL2KEAP1NFE2L2
SCHEMBL168694 0.74 CASP1 (0.42) SCN5ASCN9A
SCHEMBL9927092 0.74 SCN5A (0.36) SCN5ASCN9AAGBL2KEAP1NFE2L2
SCHEMBL27604299 0.73 KEAP1 (0.46) SCN5ASCN9AAGBL2KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012028645-A1 METHOD FOR THE PRODUCTION OF 5-FLUORO-1H-PYRAZOLO[3,4-B]PYRIDINE-3-CARBONITRILE BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-08 WO disclosed