SCHEMBL25679010

SCHEMBL25679010

c1ccc(C(c2ccccc2)N2CCn3c(nnc3-c3ccncc3)C2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.42
CYP2D6 P10635 5/20 0.41
USP2 O75604 4/20 0.41
CYP1A2 P05177 4/20 0.41
CYP2C9 P11712 4/20 0.41
CYP2C19 P33261 3/20 0.41
CYP3A4 P08684 3/20 0.41
P2RX7 Q99572 2/20 0.40
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM5 P08912 1/20 0.40
ADRA2A P08913 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
DRD1 P21728 1/20 0.40
ADRA1D P25100 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HRH1 P35367 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25679011 0.92 HPGD (0.50) HPGDCYP2D6P2RX7CHRM2CHRM4
SCHEMBL25679151 0.86 CHRM2 (0.40) HPGDCYP2D6USP2P2RX7CHRM2
SCHEMBL25679853 0.85 CHRM2 (0.49) HPGDCYP2D6USP2CYP1A2CYP2C19
SCHEMBL25679855 0.85 P2RX7 (0.49) HPGDCYP2D6CYP1A2CYP2C9CYP2C19
SCHEMBL25679957 0.84 OPRD1 (0.47) CYP3A4P2RX7OPRM1ALDH1A1NPSR1
SCHEMBL25680084 0.83 OPRD1 (0.46) CYP3A4P2RX7OPRM1ALDH1A1NPSR1
SCHEMBL25679602 0.83 OPRM1 (0.38) CYP2D6USP2CYP1A2CYP2C9CYP2C19
SCHEMBL25679141 0.82 TACR3 (0.58) CYP2D6CYP1A2CYP2C9CYP2C19P2RX7
SCHEMBL25676368 0.81 DPP4 (0.43) HPGDCYP2D6P2RX7CHRM2CHRM4
SCHEMBL25680562 0.81 ALDH1A1 (0.39) HPGDCYP2D6USP2P2RX7CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023122260-A2 INHIBITORS OF SARS-COV-2 THE TEXAS A&M UNIVERSITY SYSTEM (US) 2023-06-29 WO disclosed