SCHEMBL2574359

SCHEMBL2574359

CC1(C)Cc2cc(C(=O)O)ccc2NC1c1ccc(F)c(Nc2ccc(F)cc2Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKAG1 P54619 2/20 0.38
PRKAA1 Q13131 2/20 0.38
PRKAB1 Q9Y478 2/20 0.38
PRKAB2 O43741 1/20 0.38
PRKAA2 P54646 1/20 0.38
PRKAG3 Q9UGI9 1/20 0.38
PRKAG2 Q9UGJ0 1/20 0.38
AURKA O14965 1/20 0.38
PYGL P06737 2/20 0.37
CSNK2A1 P68400 1/20 0.34
HDAC3 O15379 1/20 0.33
RXRA P19793 1/20 0.33
HNF4A P41235 1/20 0.33
ALOX15 P16050 3/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
GALK1 P51570 1/20 0.32
PDGFRB P09619 1/20 0.32
KDR P35968 1/20 0.32
MAPK14 Q16539 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2530125 0.87 PYGL (0.43) PRKAG1PRKAA1PRKAB1PRKAB2PRKAA2
SCHEMBL2567515 0.84 KDM4E (0.37) PRKAG1PRKAA1PRKAB1PRKAB2PRKAA2
SCHEMBL2529433 0.84 PRKAG1 (0.46) PRKAG1PRKAA1PRKAB1PRKAB2PRKAA2
SCHEMBL2577051 0.83 ALDH1A1 (0.40) ALOX15ALDH1A1MAPK14BCL6BCOR
SCHEMBL2529993 0.80 TSHR (0.39) PRKAG1PRKAA1PRKAB1PRKAB2PRKAA2
SCHEMBL2529499 0.80 CYP26A1 (0.36) PRKAG1PRKAA1PRKAB1PRKAB2PRKAA2
SCHEMBL2533068 0.80 PPARG (0.46) HDAC3MAPK14
SCHEMBL2529403 0.79 HDAC8 (0.40) HDAC3ALDH1A1TSHR
SCHEMBL2574754 0.79 HCAR3 (0.35) PRKAG1PRKAA1PRKAB1PRKAB2PRKAA2
SCHEMBL2573957 0.79 IDH1 (0.38) CSNK2A1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558449-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2013-02-20 EP disclosed
WO-2011128251-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-10-20 WO disclosed