SCHEMBL25759510

SCHEMBL25759510

CCOC(=O)Cc1ccc(N)cc1S(=O)(=O)Nc1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.47
POLB P06746 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
TP53 P04637 1/20 0.46
IDH1 O75874 10/20 0.46
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23846466 0.91 LMNA (0.47) MAPTPOLBTDP1KMT2AMEN1
SCHEMBL23846511 0.89 NHERF1 (0.49) MAPTTP53IDH1KMT2AMEN1
SCHEMBL25754837 0.83 MAPT (0.58) MAPTPOLBNPSR1TDP1TP53
SCHEMBL25754913 0.83 IDH1 (0.52) MAPTTP53IDH1KMT2AMEN1
SCHEMBL25759512 0.79 MAPT (0.47) MAPTPOLBNPSR1TDP1TP53
SCHEMBL23846510 0.78 MAPT (0.44) MAPTPOLBNPSR1TDP1IDH1
SCHEMBL15647028 0.75 IDH1 (0.66) MAPTPOLBNPSR1TDP1IDH1
SCHEMBL25754797 0.74 GAA (0.50) MAPTPOLBTDP1TP53KMT2A
SCHEMBL23833760 0.74 MEN1 (0.48) MAPTNPSR1KMT2AMEN1KDM4E
SCHEMBL1354053 0.74 MAOA (0.44) MAPTKMT2AMEN1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2023-06-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF TRAP1, PINK1, TP53BP1 MAPT 89/4885POLB 1494/4885NPSR1 1552/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.