SCHEMBL257866

SCHEMBL257866

COC(C)(C)C(C)(C)OBc1ccc(CBr)cc1

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8283344 0.84 TRPA1 (0.30) TRPA1ALDH1A1TSHR
SCHEMBL10089190 0.77 CES1 (0.32) ALDH1A1
SCHEMBL9972571 0.77 ACHE (0.34) ALDH1A1TSHR
SCHEMBL10269858 0.76
SCHEMBL10193348 0.76 CA1 (0.44) ALDH1A1TSHR
SCHEMBL257867 0.73 SLC6A4 (0.39) ALDH1A1
SCHEMBL257994 0.70 SLC6A4 (0.42) ALDH1A1
SCHEMBL14232082 0.69 ENPP2 (0.34) TSHR
SCHEMBL12927941 0.69 CA1 (0.47) ALDH1A1TSHR
SCHEMBL9694556 0.67 RORC (0.39) TRPA1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2399585-A1 Boronic acids and esters as inhibitors of fatty acid amide hydrolase Infinity Pharmaceuticals, Inc. (US) 2011-12-28 EP disclosed
EP-2073816-B1 BORONIC ACIDS AND ESTERS AS INHIBITORS OF FATTY ACID AMIDE HYDROLASE INFINITY PHARMACEUTICALS INC (US) 2011-09-14 EP disclosed
WO-2009010488-A1 HETEROCYCLIC COMPOUNDS USEFUL AS MK2 INHIBITORS NOVARTIS AG (CH) 2009-01-22 WO disclosed