SCHEMBL258026

SCHEMBL258026

Oc1ccc(Br)c(F)c1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 3/20 0.40
KDM1A O60341 2/20 0.39
KCNH2 Q12809 2/20 0.39
KDM1B Q8NB78 2/20 0.39
NQO2 P16083 1/20 0.35
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
AR P10275 1/20 0.32
ALOX12 P18054 1/20 0.31
MEP1B Q16820 1/20 0.31
PIM1 P11309 1/20 0.30
ADRA2A P08913 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30
ADRA1A P35348 1/20 0.30
SNCA P37840 1/20 0.30
ADRB2 P07550 1/20 0.30
ADRA1B P35368 1/20 0.30
CES2 O00748 1/20 0.30
GALR3 O60755 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31361439 1.00 ALOX15 (0.40) ALOX15KDM1AKCNH2KDM1BNQO2
SCHEMBL855230 0.82 KDM1A (0.48) KDM1AKCNH2KDM1B
SCHEMBL29666934 0.82 KDM1A (0.48) KDM1AKCNH2KDM1B
SCHEMBL29987655 0.82 PIM1 (0.41) ALOX15ESR1ESR2ARPIM1
SCHEMBL1512796 0.82 PIM1 (0.41) ALOX15ESR1ESR2ARPIM1
SCHEMBL28694200 0.81 ALOX15 (0.39) ALOX15NQO2ESR1ESR2AR
SCHEMBL28975669 0.81 ALOX15 (0.39) ALOX15KDM1AKCNH2KDM1BNQO2
SCHEMBL30129349 0.81 ADRA2A (0.42) ALOX15KDM1AKCNH2KDM1BNQO2
SCHEMBL27949463 0.81 ALOX15 (0.39) ALOX15NQO2ESR1ESR2ALOX12
SCHEMBL4589607 0.81 ADRA2A (0.42) ALOX15KDM1AKCNH2KDM1BNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 396 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105085190-A Preparing method of 2,6-difluoro-4-bromophenol CECEP VALIANT CO LTD 2015-11-25 CN claimed
US-20260116891-A1 Oxazepin Derivative TEIJIN PHARMA LTD (JP) 2026-04-30 US disclosed
WO-2026087442-A1 AMINO-IMIDAZOLE ANTIBACTERIAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2026-04-30 WO disclosed
US-20260085064-A1 SUBSTITUTED BENZOFURANYL AND BENZOXAZOLYL COMPOUNDS AND USES THEREOF KARYOPHARM THERAPEUTICS INC (US) 2026-03-26 US disclosed
EP-4700068-A1 SILANE COMPOUND Daikin Industries, Ltd. (JP) 2026-02-25 EP disclosed
US-20260049092-A1 ANTIBACTERIAL COMPOUNDS BLACKSMITH MEDICINES INC (US) 2026-02-19 US disclosed
EP-4161931-B1 NOVEL IMIDAZOPYRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2026-02-18 EP disclosed
EP-3941919-B1 PYRIDO-PYRIMIDINONE AND PTERIDINONE COMPOUNDS AS INHIBITORS OF ENDORIBONUCLEASE INOSITOL REQUIRING ENZYME I (IRE I ALPHA) FOR THE TREATMENT OF CANCER DISEASES. GENENTECH INC (US) 2025-12-24 EP disclosed
US-12344603-B2 Pyrido-pyrimidinone and pteridinone compounds and methods of use GENENTECH, INC. (US) 2025-07-01 US disclosed
EP-4568955-A1 ANTIBACTERIAL COMPOUNDS Blacksmith Medicines, Inc. (US) 2025-06-18 EP disclosed
WO-2005077892-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2005-08-25 WO disclosed
WO-2004047751-A2 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2004-06-10 WO disclosed
EP-1214306-A1 LIQUID CRYSTAL COMPOUNDS Qinetiq Limited (GB) 2002-06-19 EP disclosed
EP-1173170-A4 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO INC (US) 2002-05-29 EP disclosed
EP-1173170-A1 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Merck & Co., Inc. (US) 2002-01-23 EP disclosed
US-6265434-B1 ANTIINFLAMMATORY AGENTS MERCK & CO., INC. 2001-07-24 US disclosed
WO-2001021606-A1 LIQUID CRYSTAL COMPOUNDS QINETIQ LIMITED (GB) 2001-03-29 WO disclosed
JP-2000309555-A PRODUCTION OF p-BROMOPHENOL COMPOUND KANTO DENKA KOGYO CO LTD 2000-11-07 JP disclosed
WO-2000059503-A1 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-10-12 WO disclosed
EP-0500210-A2 Liquid crystal compounds and compositions SANYO CHEMICAL INDUSTRIES, LTD. (JP) 1992-08-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260049092-A1 ANTIBACTERIAL COMPOUNDS H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, CBR1, FPR1 ALOX15 1523/4885KDM1A 2592/4885KCNH2 531/4885
US-12344603-B2 Pyrido-pyrimidinone and pteridinone compounds and methods of use TYMP, TYMS, DPYD ALOX15 1722/4885KDM1A 2560/4885KCNH2 4574/4885
US-20260116891-A1 Oxazepin Derivative HCRTR2, HCRTR1, OXTR ALOX15 915/4885KDM1A 2119/4885KCNH2 600/4885
US-20260085064-A1 SUBSTITUTED BENZOFURANYL AND BENZOXAZOLYL COMPOUNDS AND USES THEREOF BCL6, MALT1, BCL6B ALOX15 1359/4885KDM1A 581/4885KCNH2 401/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.