Phenolsulphonic Acid

Phenolsulphonic Acid

SCHEMBL2581592

O.O=S(=O)(O)c1ccccc1O

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Phenolsulphonic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR known ✓ P00533 1/20 0.43
PIK3CA known ✓ P42336 1/20 0.43
AURKA O14965 1/20 0.44
AURKB Q96GD4 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
TSHR P16473 1/20 0.44
MYC P01106 1/20 0.44
CDK2 P24941 1/20 0.43
CA2 P00918 3/20 0.43
CA4 P22748 3/20 0.43
LMNA P02545 2/20 0.43
HPGD P15428 2/20 0.43
HIF1A Q16665 2/20 0.43
HSD17B10 Q99714 2/20 0.43
POLB P06746 2/20 0.43
CA12 O43570 2/20 0.43
CA5A P35218 2/20 0.43
CA14 Q9ULX7 2/20 0.43
CA5B Q9Y2D0 2/20 0.43
TDP1 Q9NUW8 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenolsulphonic Acid SCHEMBL9169950 1.00 AURKA (0.44) AURKAAURKBSMN1; SMN2TSHRMYC
Phenolsulphonic Acid SCHEMBL28340891 1.00 AURKA (0.44) AURKAAURKBSMN1; SMN2TSHRMYC
Phenolsulphonic Acid SCHEMBL2914071 0.98 AURKA (0.43) AURKAAURKBSMN1; SMN2TSHRMYC
Phenolsulphonic Acid SCHEMBL28907966 0.98 AURKA (0.43) AURKAAURKBSMN1; SMN2TSHRMYC
Phenolsulphonic Acid SCHEMBL18274 0.97 SMN1; SMN2 (0.46) AURKAAURKBSMN1; SMN2TSHRMYC
Phenolsulphonic Acid SCHEMBL29449532 0.97 SMN1; SMN2 (0.46) AURKAAURKBSMN1; SMN2TSHRMYC
Phenolsulphonic Acid SCHEMBL11154671 0.97 SMN1; SMN2 (0.46) AURKAAURKBSMN1; SMN2TSHRMYC
Phenolsulphonic Acid SCHEMBL2519919 0.95 SMN1; SMN2 (0.50) AURKAAURKBSMN1; SMN2TSHRMYC
Phenolsulphonic Acid SCHEMBL812225 0.95 AURKA (0.44) AURKAAURKBSMN1; SMN2TSHRMYC
Phenolsulphonic Acid SCHEMBL10587629 0.95 SMN1; SMN2 (0.50) AURKAAURKBSMN1; SMN2TSHRMYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118450802-A Viral infection suppressing member 积水化学工业株式会社 2024-08-06 CN disclosed
WO-2023171557-A1 VIRAL INFECTION-INHIBITING MEMBER 積水化学工業株式会社 2023-09-14 WO disclosed
EP-2563797-A2 METHOD FOR PRODUCING MIXTURES OF ALKYLPHOSPHONOUS ACID SALTS AND DIALKYLPHOSPHINIC ACID SALTS Clariant Finance (BVI) Limited (VG) 2013-03-06 EP disclosed
EP-2563798-A2 METHOD FOR PRODUCING ALKYLPHOSPHONOUS ACID SALTS Clariant Finance (BVI) Limited (VG) 2013-03-06 EP disclosed
WO-2011134621-A2 METHOD FOR PRODUCING ALKYLPHOSPHONOUS ACID SALTS CLARIANT INTERNATIONAL LTD (CH) 2011-11-03 WO disclosed
WO-2011134620-A2 METHOD FOR PRODUCING MIXTURES OF ALKYLPHOSPHONOUS ACID SALTS AND DIALKYLPHOSPHINIC ACID SALTS CLARIANT INTERNATIONAL LTD (CH) 2011-11-03 WO disclosed
EP-0268374-B1 Method for treating fibrous polyamide materials with divalent metal salts of sulfonated novolak resins. MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1993-02-10 EP disclosed
US-5098774-A Stain resistant finishes CHANG JOHN C (US) 1992-03-24 US disclosed
EP-0268374-A2 Method for treating fibrous polyamide materials with divalent metal salts of sulfonated novolak resins. MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1988-05-25 EP disclosed