SCHEMBL25839066

SCHEMBL25839066

Cc1cnc2[nH]cc(Oc3ccncc3)c2c1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.41
PIK3CA P42336 1/20 0.41
SLC2A1 P11166 1/20 0.41
AXL P30530 1/20 0.40
NTRK1 P04629 8/20 0.40
CYP3A4 P08684 4/20 0.39
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 1/20 0.37
NEK1 Q96PY6 1/20 0.36
AAK1 Q2M2I8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24565966 0.77 KIT (0.48) KITCYP3A4CYP2C9CYP2C19AAK1
SCHEMBL17952128 0.75 NTRK1 (0.62) KITPIK3CASLC2A1AXLNTRK1
SCHEMBL22049447 0.72 CYP2C9 (0.36) KITCYP3A4CYP2C9CYP2C19AAK1
SCHEMBL27920535 0.71 SLC22A6 (0.45) KITAXLCYP3A4CYP2C9CYP2C19
SCHEMBL25781685 0.70 NTRK1 (0.47) KITPIK3CASLC2A1AXLNTRK1
SCHEMBL7921128 0.69 MET (0.46) AXLCYP3A4CYP2C9CYP2C19
SCHEMBL13199598 0.66 CYP3A4 (0.44) KITCYP3A4CYP2C9CYP2C19
SCHEMBL15154998 0.66 GSK3B (0.56) KITNTRK1CYP3A4CYP2C9CYP2C19
SCHEMBL21902710 0.66 CYP2C19 (0.40) CYP3A4CYP2C9CYP2C19
SCHEMBL31228005 0.66 BRD4 (0.54) KITAXLCYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed