SCHEMBL25839071

SCHEMBL25839071

Cc1cnc2[nH]cc(N(C)C)c2c1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 1/20 0.40
CYP3A4 P08684 5/20 0.36
CYP2C19 P33261 4/20 0.36
CYP2C9 P11712 4/20 0.36
MAPK8 P45983 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK10 P53779 1/20 0.36
BRAF P15056 1/20 0.36
NTRK1 P04629 1/20 0.35
EDNRA P25101 1/20 0.33
CAMKK2 Q96RR4 1/20 0.33
KIT P10721 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16320524 0.81 AXL (0.36) MAP3K11CYP3A4CYP2C19BRAFCAMKK2
SCHEMBL26018150 0.81 BRAF (0.40) MAP3K11CYP3A4CYP2C9MAPK8MAPK9
SCHEMBL1772956 0.81 MAP3K11 (0.39) MAP3K11CYP3A4MAPK8MAPK9MAPK10
SCHEMBL7921128 0.77 MET (0.46) CYP3A4CYP2C19CYP2C9
SCHEMBL7965037 0.75 CYP3A4 (0.44) CYP3A4CYP2C19CYP2C9KIT
SCHEMBL1772835 0.74 ALDH1A1 (0.43) MAP3K11BRAF
SCHEMBL13199598 0.74 CYP3A4 (0.44) CYP3A4CYP2C19CYP2C9BRAFKIT
SCHEMBL31228005 0.74 BRD4 (0.54) CYP3A4CYP2C19CYP2C9MAPK8KIT
SCHEMBL21902710 0.74 CYP2C19 (0.40) MAP3K11CYP3A4CYP2C19CYP2C9BRAF
SCHEMBL15154998 0.74 GSK3B (0.56) MAP3K11CYP3A4CYP2C19CYP2C9NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed