SCHEMBL2584063

SCHEMBL2584063

CS(=O)(=O)O[C@@H]1[C@@H](O)[C@H](n2cnc3ncnc-3c2Cl)O[C@@H]1CO

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HTT P42858 2/20 0.38
BLM P54132 2/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
ADORA3 P0DMS8 2/20 0.37
DPP4 P27487 1/20 0.37
MEN1 O00255 1/20 0.37
SLC28A1 O00337 1/20 0.37
MAP3K7 O43318 1/20 0.37
SLC28A2 O43868 1/20 0.37
GAPDH P04406 1/20 0.37
MAPK1 P28482 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA2B P29275 1/20 0.37
ADORA1 P30542 1/20 0.37
STAT6 P42226 1/20 0.37
PI4KA P42356 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2584222 0.87 ADORA1 (0.37) SMN1; SMN2ALDH1A1HTTBLMKDM4E
SCHEMBL2579342 0.86 SMN1; SMN2 (0.38) SMN1; SMN2ALDH1A1HTTBLMKDM4E
SCHEMBL2584026 0.85 ADK (0.36) SLC28A2LMNATP53HPGD
SCHEMBL2578109 0.81 SLC29A1 (0.53) SMN1; SMN2ALDH1A1HTTBLMADORA3
SCHEMBL6886934 0.80 SLC29A1 (0.51) SMN1; SMN2ADORA3DPP4MEN1SLC28A1
SCHEMBL2584815 0.80 HSPA5 (0.37) ALDH1A1HTTBLMKDM4ESLC28A2
SCHEMBL2587219 0.79 HSPA8 (0.34) SLC28A2SLC29A1
SCHEMBL2579190 0.78 LMNA (0.51) SMN1; SMN2ALDH1A1LMNATP53
SCHEMBL6885472 0.75 SLC29A1 (0.52) SMN1; SMN2ADORA3DPP4MEN1SLC28A1
SCHEMBL6889026 0.75 LMNA (0.69) ALDH1A1ADORA3MEN1MAPK1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10100076-B2 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation GILEAD PHARMASSET LLC (US) 2018-10-16 US disclosed
US-20140057863-A1 MODIFIED NUCLEOSIDES FOR THE TREATMENT OF VIRAL INFECTIONS AND ABNORMAL CELLULAR PROLIFERATION GILEAD SCIENCES, INC. (US) 2014-02-27 US disclosed
EP-2251015-B1 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation GILEAD PHARMASSET LLC (US) 2013-02-20 EP disclosed
US-20110269707-A1 Modified nucleosides for the treatment of viral infections and abnormal cellullar proliferation PHARMASSET, INC. 2011-11-03 US disclosed
EP-2251015-A1 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation Pharmasset, Inc. (US) 2010-11-17 EP disclosed
US-20030087873-A1 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation PHARMASSET, INC. 2003-05-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140057863-A1 MODIFIED NUCLEOSIDES FOR THE TREATMENT OF VIRAL INFECTIONS AND ABNORMAL CELLULAR PROLIFERATION SLC29A1, PNP, SLC29A2 SMN1; SMN2 214/4885ALDH1A1 1466/4885HTT 4480/4885
US-20110269707-A1 Modified nucleosides for the treatment of viral infections and abnormal cellullar proliferation PNP, ALPP, XDH SMN1; SMN2 676/4885ALDH1A1 2416/4885HTT 4766/4885
US-10100076-B2 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation SLC29A1, SLC29A2, PNP SMN1; SMN2 63/4885ALDH1A1 1128/4885HTT 4514/4885
US-20030087873-A1 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation SLC29A1, PNP, SLC29A2 SMN1; SMN2 244/4885ALDH1A1 1367/4885HTT 4574/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.