SCHEMBL258432

SCHEMBL258432

CCOC(=O)c1sc2ncccc2c1N

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.65
CHUK O15111 1/20 0.65
LIMK1 P53667 1/20 0.65
KDM4E B2RXH2 7/20 0.64
MAPT P10636 5/20 0.64
NPC1 O15118 3/20 0.64
RAB9A P51151 3/20 0.64
MEN1 O00255 1/20 0.64
POLB P06746 1/20 0.64
NFKB1 P19838 1/20 0.64
NFKB2 Q00653 1/20 0.64
KMT2A Q03164 1/20 0.64
RELA Q04206 1/20 0.64
HPGD P15428 6/20 0.62
SMN1; SMN2 Q16637 4/20 0.62
ALDH1A1 P00352 6/20 0.52
GAA P10253 3/20 0.52
HSD17B10 Q99714 3/20 0.52
GLA P06280 2/20 0.52
CASP1 P29466 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30338754 1.00 IKBKB (0.65) IKBKBCHUKLIMK1KDM4EMAPT
SCHEMBL719584 0.86 KDM4E (0.58) IKBKBCHUKLIMK1KDM4EMAPT
SCHEMBL2896095 0.86 IKBKB (0.68) IKBKBCHUKLIMK1KDM4EMAPT
SCHEMBL16475087 0.84 KDM4E (0.57) IKBKBCHUKLIMK1KDM4EMAPT
SCHEMBL1266041 0.83 KDM4E (0.56) IKBKBCHUKLIMK1KDM4EMAPT
SCHEMBL22638989 0.82 IKBKB (0.63) IKBKBCHUKLIMK1KDM4EMAPT
SCHEMBL9541091 0.82 IKBKB (0.63) IKBKBCHUKLIMK1KDM4EMAPT
SCHEMBL29707339 0.81 KDM4E (0.70) IKBKBLIMK1KDM4EMAPTNPC1
SCHEMBL3494383 0.81 KDM4E (0.70) IKBKBLIMK1KDM4EMAPTNPC1
SCHEMBL16475088 0.80 KDM4E (0.61) IKBKBCHUKLIMK1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 151 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12297209-B2 Benzodiazepine derivatives as RSV inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2025-05-13 US disclosed
US-12268694-B2 Combination pharmaceutical agents as RSV inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2025-04-08 US disclosed
US-20240360155-A1 Benzodiazepine Derivatives as RSV Inhibitors ENANTA PHARM INC (US) 2024-10-31 US disclosed
US-11952389-B2 Benzodiazepine derivatives as RSV inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2024-04-09 US disclosed
EP-3687543-B1 COMBINATIONS OF PHARMACEUTICAL AGENTS AS RSV INHIBITORS ENANTA PHARM INC (US) 2024-03-20 EP disclosed
US-20230087410-A1 BENZODIAZEPINE DERIVATIVES AS RSV INHIBITORS ENANTA PHARM INC (US) 2023-03-23 US disclosed
US-20230084927-A1 GLUCOSE UPTAKE INHIBITORS AND USES THEREOF METABOMED LTD. (IL) 2023-03-16 US disclosed
US-20220323460-A1 COMBINATION PHARMACEUTICAL AGENTS AS RSV INHIBITORS ENANTA PHARM INC (US) 2022-10-13 US disclosed
EP-4058027-A1 GLUCOSE UPTAKE INHIBITORS AND USES THEREOF Metabomed Ltd (IL) 2022-09-21 EP disclosed
US-11390631-B1 Benzodiazepine derivatives as RSV inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2022-07-19 US disclosed
US-20040009978-A1 Fused heteroaryl derivatives ASTELLAS PHARMA INC. (JP) 2004-01-15 US disclosed
US-20030236271-A1 Fused heteroaryl derivatives ASTELLAS PHARMA INC. (JP) 2003-12-25 US disclosed
US-6608056-B1 Phosphatidylinositol 3-kinase inhibitors and carcinostatic agents YAMANOUCHI PHARMACEUTICAL CO., LTD (JP) 2003-08-19 US disclosed
US-6608053-B2 Phosphatidylinositol 3-kinase (PI3K) inhibitors/anticancer agents such as N-(2-(3-benzenesulfonylaminophenyl)-4-morphoniloquinazolin-6-yl)acetamide YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2003-08-19 US disclosed
EP-1277738-A1 CONDENSED HETEROARYL DERIVATIVES YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 2003-01-22 EP disclosed
US-20020151544-A1 Fused heteroaryl derivatives ASTELLAS PHARMA INC. (JP) 2002-10-17 US disclosed
US-6133275-A ALPHA 1 ADRENORECEPTOR ANTAGONISTS; TREATING BENIGN PROSTATIC HYPERPLASIA AND OTHER UROLOGICAL DISEASES E.G., BLADDER OUTLET OBSTRUCTION), NEUROGENIC BLADDER AND GYNECOLOGICAL SYNDROMES, E.G., DYSMENORRHEA; UTERINE MUSCLE RELAXANTS ABBOTT LABORATORIES (US) 2000-10-17 US disclosed
EP-0004319-B1 N-(PYRIDOTHIENOPYRAZOL) AMIDES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM E.I. DU PONT DE NEMOURS AND COMPANY (US) 1981-08-05 EP disclosed
US-4220776-A TREATMENT OF RHINOVIRAL INFECTIONS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1980-09-02 US disclosed
EP-0004319-A1 N-(pyridothienopyrazol) amides, process for their preparation and pharmaceutical compositions containing them E.I. DU PONT DE NEMOURS AND COMPANY (US) 1979-10-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030236271-A1 Fused heteroaryl derivatives PIK3CD, PIK3R3, PIK3C2A IKBKB 339/4885CHUK 37/4885LIMK1 1080/4885
US-20240360155-A1 Benzodiazepine Derivatives as RSV Inhibitors GABRA5, GABRA1, GABBR2 IKBKB 598/4885CHUK 130/4885LIMK1 4734/4885
US-20040009978-A1 Fused heteroaryl derivatives PIK3CD, PIK3R3, PIK3C2A IKBKB 339/4885CHUK 37/4885LIMK1 1080/4885
US-11952389-B2 Benzodiazepine derivatives as RSV inhibitors GABRA5, GABRA1, GABBR2 IKBKB 598/4885CHUK 130/4885LIMK1 4734/4885
US-11390631-B1 Benzodiazepine derivatives as RSV inhibitors GABRA5, GABRA1, GABBR2 IKBKB 598/4885CHUK 130/4885LIMK1 4734/4885
US-12297209-B2 Benzodiazepine derivatives as RSV inhibitors GABRA5, GABRA1, GABBR2 IKBKB 598/4885CHUK 130/4885LIMK1 4734/4885
US-20220323460-A1 COMBINATION PHARMACEUTICAL AGENTS AS RSV INHIBITORS SERPINB1, FURIN, HIF1AN IKBKB 186/4885CHUK 11/4885LIMK1 4408/4885
US-20230087410-A1 BENZODIAZEPINE DERIVATIVES AS RSV INHIBITORS GABRA5, GABRA1, GABBR2 IKBKB 598/4885CHUK 130/4885LIMK1 4734/4885
US-20020151544-A1 Fused heteroaryl derivatives PIK3CD, PIK3R3, PIK3C2A IKBKB 339/4885CHUK 37/4885LIMK1 1080/4885
US-12268694-B2 Combination pharmaceutical agents as RSV inhibitors ACE, ACE2, SPCS3 IKBKB 315/4885CHUK 41/4885LIMK1 4362/4885
US-20230084927-A1 GLUCOSE UPTAKE INHIBITORS AND USES THEREOF SLC2A4, SLC2A1, SLC2A2 IKBKB 1267/4885CHUK 408/4885LIMK1 3294/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.