SCHEMBL25859255

SCHEMBL25859255

CC#Cc1ccc(-c2nnc(N)c3ccccc23)c(OCOCC)c1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP1B1 Q16678 1/20 0.33
NCF1 P14598 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 2/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
CACNA2D1 P54289 2/20 0.30
CRHR1 P34998 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25860910 0.88 NCF1 (0.33) NCF1KDM4EMAPTMEN1ALDH1A1
SCHEMBL25858870 0.85 ALDH1A1 (0.38) CYP1A1CYP1A2CYP1B1KDM4EMAPT
SCHEMBL31314270 0.80 ALOX5AP (0.41) NCF1MAPTMEN1ALDH1A1HTT
SCHEMBL25857192 0.80 DHFR (0.37) CYP1A2NCF1KDM4EMAPTALDH1A1
SCHEMBL25859018 0.79 CACNA2D1 (0.34) KMT2ACACNA2D1
SCHEMBL25856433 0.78 KDM4E (0.41) CYP1A1CYP1A2CYP1B1KDM4EMEN1
SCHEMBL25857355 0.76 PIP4K2A (0.30)
SCHEMBL25859817 0.76
SCHEMBL25861428 0.76 ALDH1A1 (0.37) KDM4EMAPTALDH1A1HTTNPSR1
SCHEMBL30517778 0.75 GRM5 (0.35) KDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed