SCHEMBL2586009

SCHEMBL2586009

Cc1cc(C(=O)N2CCc3onc(C(=O)NCCN4CCCC4)c3C2)ccc1Br

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 10/20 0.53
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
POLB P06746 1/20 0.43
NPSR1 Q6W5P4 1/20 0.41
EEF2K O00418 1/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 2/20 0.40
HPGD P15428 2/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2588891 0.93 HSP90AA1 (0.62) HSP90AA1HDAC3HDAC4HDAC1HDAC7
SCHEMBL2576088 0.89 HSP90AA1 (0.54) HSP90AA1HDAC3HDAC4HDAC1HDAC7
SCHEMBL4267339 0.82 HSP90AA1 (0.46) HSP90AA1HDAC3HDAC4HDAC1HDAC7
SCHEMBL2579235 0.81 HSP90AA1 (0.51) HSP90AA1HDAC3HDAC4HDAC1HDAC7
SCHEMBL7978285 0.76 NPSR1 (0.65) HDAC2HDAC8HDAC6POLBNPSR1
SCHEMBL5528804 0.74 HPGD (0.40) HSP90AA1KMT2AHPGDALDH1A1NPC1
SCHEMBL2584836 0.73 HSP90AA1 (0.49) HSP90AA1HDAC3HDAC4HDAC1HDAC7
SCHEMBL2586692 0.72 RAB9A (0.48) HSP90AA1EEF2KKMT2AGAAHPGD
SCHEMBL2587431 0.71 HSP90AA1 (0.46) HSP90AA1KMT2AGAAALDH1A1KDM4E
SCHEMBL2579206 0.71 HSP90AA1 (0.52) HSP90AA1HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US claimed
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US disclosed