SCHEMBL258716

SCHEMBL258716

Nc1ccc(CNC(=O)O)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.62
CYP2C19 P33261 2/20 0.62
CYP1A2 P05177 1/20 0.62
CYP2D6 P10635 1/20 0.62
TSHR P16473 1/20 0.62
PPID Q08752 3/20 0.56
PPIB P23284 2/20 0.56
PPIA P62937 1/20 0.56
PPIG Q13427 1/20 0.56
EPHX2 P34913 1/20 0.54
EPHX1 P07099 1/20 0.53
TPSAB1 Q15661 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ITGB1 P05556 2/20 0.49
ITGA5 P08648 2/20 0.49
KMT2A Q03164 2/20 0.47
KDM4E B2RXH2 2/20 0.47
MAPT P10636 1/20 0.47
HIF1A Q16665 1/20 0.47
SLC22A6 Q4U2R8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7441659 0.98 CYP2C9 (0.60) CYP2C9CYP2C19CYP1A2CYP2D6TSHR
SCHEMBL20497326 0.94 CYP1A2 (0.56) CYP2C9CYP2C19CYP1A2CYP2D6TSHR
SCHEMBL11533429 0.91 CYP2C9 (0.65) CYP2C9CYP2C19CYP1A2CYP2D6TSHR
Alanine SCHEMBL22445734 0.87 ITGB1 (0.51) CYP2C9CYP2C19CYP1A2CYP2D6TSHR
SCHEMBL15939528 0.86 PPID (0.65) CYP2C9CYP2C19PPIDPPIBPPIA
SCHEMBL20705214 0.85 CYP2C19 (0.61) CYP2C9CYP2C19CYP1A2CYP2D6TSHR
SCHEMBL972153 0.85 PPID (0.55) CYP2C9CYP2C19CYP1A2CYP2D6TSHR
SCHEMBL4738233 0.84 CYP2C9 (0.85) CYP2C9CYP2C19CYP1A2CYP2D6TSHR
SCHEMBL1919932 0.84 EPHX2 (0.53) CYP2C9CYP2C19CYP1A2CYP2D6TSHR
SCHEMBL8245710 0.84 CYP2C9 (0.68) CYP2C9CYP2C19CYP1A2CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 987 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026105061-A1 ANTIBODY-DRUG CONJUGATES THAT BIND CDCP1 AND USES THEREOF PHEON THERAPEUTICS LTD (GB) 2026-05-21 WO claimed
US-12606830-B2 Protected antibody-drug and aptamer-drug conjugates KOSAK KENNETH MICHAEL (US) 2026-04-21 US claimed
US-20260027220-A1 EPHA2 BCL-XL INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE THEREOF NOVARTIS AG (CH) 2026-01-29 US claimed
US-20260027147-A1 EXTRACELLULAR VESICLE-ASO CONSTRUCTS TARGETING CEBP/BETA LONZA SALES AG (CH) 2026-01-29 US claimed
EP-4676540-A1 PANRAS INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE THEREOF Novartis AG (CH) 2026-01-14 EP claimed
US-20250387504-A1 ANTIBODY-DRUG CONJUGATES OF ANTINEOPLASTIC COMPOUNDS AND METHODS OF USE THEREOF NOVARTIS AG (CH) 2025-12-25 US claimed
US-20250382613-A1 METHODS OF USING EXTRACELLULAR VESICLE-ASO TARGETING STAT6 LONZA SALES AG (CH) 2025-12-18 US claimed
US-20250339547-A1 MET BCL-XL INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE THEREOF NOVARTIS AG (CH) 2025-11-06 US claimed
EP-4642491-A1 METHOD FOR GLYCOPROTEIN MODIFICATION Honeybear Biosciences Inc. (TW) 2025-11-05 EP claimed
WO-2025202361-A1 ANTI-GPC1 ANTIBODIES AND USES THEREOF ADCENDO APS (DK) 2025-10-02 WO claimed
EP-2710024-A2 OSW-1 ANALOGS AND CONJUGATES, AND USES THEREOF President and Fellows of Harvard College (US) 2014-03-26 EP claimed
EP-1912677-B1 PSMA antibody-drug conjugates PSMA DEV COMPANY L L C (US) 2013-10-02 EP claimed
EP-2326350-B1 COMPOUNDS FOR KILLING PSMA-EXPRESSING, TAXANE-RESISTANT CANCER CELLS PSMA DEV COMPANY L L C (US) 2013-09-04 EP claimed
WO-2012159027-A2 OSW-1 ANALOGS AND CONJUGATES, AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2012-11-22 WO claimed
EP-2326350-A2 METHODS FOR KILLING PSMA-EXPRESSING, TAXANE-RESISTANT CANCER CELLS Psma Development Company, L.L.C. (US) 2011-06-01 EP claimed
WO-2010027513-A2 METHODS FOR KILLING PSMA-EXPRESSING, TAXANE-RESISTANT CANCER CELLS PSMA DEVELOPMENT COMPANY, LLC (US) 2010-03-11 WO claimed
EP-1912677-A2 PSMA ANTIBODY-DRUG CONJUGATES Psma Development Company, L.L.C. (US) 2008-04-23 EP claimed
WO-2007002222-A2 PSMA ANTIBODY-DRUG CONJUGATES PSMA DEVELOPMENT COMPANY, LLC (US) 2007-01-04 WO claimed
US-6214345-B1 ANTITUMOR AGENTS; DRUG CONJUGATES WHICH ARE SELECTIVELY ACTIVATIBLE AT THE SITE OF THE TUMOR BRISTOL-MYERS SQUIBB CO. 2001-04-10 US claimed
US-5480989-A Carbamates of rapamycin AMERICAN HOME PRODUCTS CORPORATION (US) 1996-01-02 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260027220-A1 EPHA2 BCL-XL INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE THEREOF EPHA2, EPHA1, EPHB1 CYP2C9 2939/4885CYP2C19 3919/4885CYP1A2 3146/4885
US-20250387504-A1 ANTIBODY-DRUG CONJUGATES OF ANTINEOPLASTIC COMPOUNDS AND METHODS OF USE THEREOF BID, BCL2, MCL1 CYP2C9 3660/4885CYP2C19 4171/4885CYP1A2 3981/4885
US-20250339547-A1 MET BCL-XL INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE THEREOF MET, BCL3, BCL9 CYP2C9 2470/4885CYP2C19 3055/4885CYP1A2 4499/4885
US-20250382613-A1 METHODS OF USING EXTRACELLULAR VESICLE-ASO TARGETING STAT6 STAT6, EXOSC5, STAT5B CYP2C9 4881/4885CYP2C19 4885/4885CYP1A2 4884/4885
US-20260027147-A1 EXTRACELLULAR VESICLE-ASO CONSTRUCTS TARGETING CEBP/BETA CEBPZ, OSBP, DIS3 CYP2C9 4821/4885CYP2C19 4884/4885CYP1A2 4876/4885
US-12606830-B2 Protected antibody-drug and aptamer-drug conjugates PABPC1, PABPC4, ABCG2 CYP2C9 2431/4885CYP2C19 3366/4885CYP1A2 3519/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.