SCHEMBL25877820

SCHEMBL25877820

Cc1ccc(OCC(C)(C)O)cc1-c1ccnc(N)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 4/20 0.43
PDE2A O00408 4/20 0.41
PDE10A Q9Y233 4/20 0.41
GSK3B P49841 1/20 0.40
AAK1 Q2M2I8 2/20 0.38
PIK3CD O00329 4/20 0.38
PIK3CB P42338 4/20 0.38
PIK3CG P48736 4/20 0.38
ABL1 P00519 2/20 0.37
S1PR1 P21453 2/20 0.37
MCHR1 Q99705 1/20 0.37
PIM1 P11309 1/20 0.36
CDK9 P50750 1/20 0.36
DYRK2 Q92630 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
MTOR P42345 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23956537 0.86 DYRK1A (0.41) DYRK1APDE2APDE10AGSK3BAAK1
SCHEMBL22272533 0.81 DYRK1A (0.43) DYRK1AGSK3BAAK1ABL1S1PR1
SCHEMBL22918783 0.80 NOS3 (0.55) DYRK1APDE2APDE10AAAK1S1PR1
SCHEMBL29615423 0.80 NOS3 (0.55) DYRK1APDE2APDE10AAAK1S1PR1
SCHEMBL25877728 0.79 DYRK1A (0.64) DYRK1AGSK3BAAK1ABL1PIM1
SCHEMBL25877903 0.79 DYRK1A (0.49) DYRK1AGSK3BAAK1ABL1S1PR1
SCHEMBL22272941 0.78 MAOA (0.45) DYRK1AGSK3BAAK1ABL1S1PR1
SCHEMBL22272939 0.78 DYRK1A (0.44) DYRK1AGSK3BAAK1ABL1S1PR1
SCHEMBL30091626 0.78 DYRK1A (0.44) DYRK1AGSK3BAAK1ABL1S1PR1
SCHEMBL23956533 0.78 PDE2A (0.45) DYRK1APDE2APDE10AGSK3BAAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138433-A2 AMIDE COMPOUND HAVING RIPK1 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR, AND USE THEREOF 中国科学院上海药物研究所 2023-07-27 WO disclosed