SCHEMBL2589640

SCHEMBL2589640

COC(=O)C(O)c1c(C)c(S(=O)(=O)Cc2ccc(F)cc2)c2ccccn12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 6/20 0.55
HCRTR1 O43613 5/20 0.55
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.39
HTT P42858 1/20 0.39
HSD17B10 Q99714 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAPT P10636 4/20 0.38
POLB P06746 2/20 0.38
THRB P10828 1/20 0.38
LMNA P02545 1/20 0.38
CA12 O43570 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2592298 0.89 HCRTR2 (0.45) HCRTR2HCRTR1ALDH1A1KDM4EHPGD
SCHEMBL4635350 0.85 HTR6 (0.41) HCRTR2HCRTR1ALDH1A1KDM4EHPGD
SCHEMBL2589762 0.80 HCRTR2 (0.57) HCRTR2HCRTR1ALDH1A1KDM4EHPGD
SCHEMBL2588741 0.80 HCRTR2 (0.71) HCRTR2HCRTR1ALDH1A1KDM4EHPGD
SCHEMBL2594270 0.76 HCRTR2 (0.75) HCRTR2HCRTR1ALDH1A1HPGDSMN1; SMN2
SCHEMBL2586420 0.72 HCRTR2 (0.54) HCRTR2HCRTR1ALDH1A1KDM4EHPGD
SCHEMBL7709453 0.71 HCRTR2 (1.00) HCRTR2HCRTR1ALDH1A1L3MBTL1MAPT
SCHEMBL7710901 0.70 HCRTR2 (1.00) HCRTR2HCRTR1ALDH1A1NPSR1L3MBTL1
SCHEMBL4635361 0.69 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHTTHSD17B10
SCHEMBL2589693 0.69 HCRTR2 (0.47) HCRTR2HCRTR1ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011138266-A1 INDOLIZINE AND IMIDAZOPYRIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS EVOTEC AG (DE) 2011-11-10 WO disclosed
WO-2011138266-A1 INDOLIZINE AND IMIDAZOPYRIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS EVOTEC AG (DE) 2011-11-10 WO disclosed