SCHEMBL2589797

SCHEMBL2589797

O=C(NC1CCN(Cc2ccccc2)C1)c1noc2ccncc12

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.55
DRD2 P14416 11/20 0.53
DRD4 P21917 11/20 0.53
MCHR1 Q99705 1/20 0.52
HDAC3 O15379 1/20 0.51
HDAC4 P56524 1/20 0.51
HDAC7 Q8WUI4 1/20 0.51
HDAC9 Q9UKV0 1/20 0.51
HDAC5 Q9UQL6 1/20 0.51
NCOR2 Q9Y618 1/20 0.51
SIGMAR1 Q99720 2/20 0.50
WNT1 P04628 1/20 0.49
DYRK1A Q13627 1/20 0.49
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2580912 0.88 TEAD1 (0.54) ROCK2DRD2DRD4HDAC3HDAC4
SCHEMBL7694198 0.74 DRD2 (0.85) DRD2DRD4MCHR1SIGMAR1
SCHEMBL7694199 0.74 DRD2 (0.85) DRD2DRD4MCHR1SIGMAR1
SCHEMBL239528 0.73 DRD4 (0.71) DRD2DRD4MCHR1SIGMAR1KMT2A
SCHEMBL239527 0.73 DRD4 (0.71) DRD2DRD4MCHR1SIGMAR1KMT2A
SCHEMBL19317742 0.73 SMYD3 (0.69) MEN1ALDH1A1KMT2A
SCHEMBL19614234 0.72 DRD4 (0.70) DRD2DRD4MCHR1SIGMAR1KMT2A
SCHEMBL20183285 0.72 DRD4 (0.70) DRD2DRD4MCHR1SIGMAR1KMT2A
SCHEMBL17961749 0.72 DRD4 (0.70) DRD2DRD4MCHR1SIGMAR1KMT2A
SCHEMBL7656471 0.72 SIGMAR1 (0.65) ROCK2DRD2DRD4SIGMAR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US disclosed