SCHEMBL2591352

SCHEMBL2591352

Nc1nccc(Oc2cc(F)ccc2F)c1I

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MET P08581 12/20 0.45
KDR P35968 5/20 0.43
MAP4K4 O95819 1/20 0.36
RET P07949 1/20 0.35
KIT P10721 1/20 0.35
PDGFRA P16234 1/20 0.35
FLT3 P36888 1/20 0.35
TRPA1 O75762 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27929011 0.84 MEN1 (0.46) METKDRMAP4K4
SCHEMBL2591537 0.82 MET (0.41) METKDRMAP4K4RETKIT
SCHEMBL25362099 0.79 MET (0.48) METKDRMAP4K4RETKIT
SCHEMBL31007081 0.77 MET (0.39) METKDRKITFLT3
SCHEMBL12384866 0.74 MET (0.47) METKDRRETKITPDGFRA
SCHEMBL2591029 0.74 MET (0.39) METKDR
SCHEMBL9487857 0.74 CA3 (0.46) TRPA1
SCHEMBL1137074 0.72 HSPB1 (0.49) METKDR
SCHEMBL30495857 0.72 HSPB1 (0.49) METKDR
SCHEMBL11933610 0.70 LMNA (0.45) METKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8569319-B2 Pyridone amides and analogs exhibiting anti-cancer and anti-proliferative activities Deciphera Pharmaceuticals, LLS (US) 2013-10-29 US disclosed
EP-2563773-A1 PYRIDONE AMIDES AND ANALOGS EXHIBITING ANTI-CANCER AND ANTI-PROLIFERATIVE ACTIVITES Deciphera Pharmaceuticals, LLC (US) 2013-03-06 EP disclosed
US-20120172382-A1 PYRIDONE AMIDES AND ANALOGS EXHIBITING ANTI-CANCER AND ANTI-PROLIFERATIVE ACTIVITIES DECIPHERA PHARMACEUTICALS, LLC. (US) 2012-07-05 US disclosed
WO-2011139891-A1 PYRIDONE AMIDES AND ANALOGS EXHIBITING ANTI-CANCER AND ANTI-PROLIFERATIVE ACTIVITES DECIPHERA PHARMACEUTICALS, LLC (US) 2011-11-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120172382-A1 PYRIDONE AMIDES AND ANALOGS EXHIBITING ANTI-CANCER AND ANTI-PROLIFERATIVE ACTIVITIES MKI67, TYMP, CCNA1 MET 2197/4885KDR 2384/4885MAP4K4 614/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.