SCHEMBL25925229

SCHEMBL25925229

CN1CCC(n2cc(-c3cn(S(=O)(=O)c4ccccc4)c4ncc(Br)nc34)cn2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.39
ACVR1 Q04771 2/20 0.39
BMPR1A P36894 1/20 0.39
ACVRL1 P37023 1/20 0.39
MAP3K7 O43318 6/20 0.38
TAB1 Q15750 6/20 0.38
IKBKE Q14164 1/20 0.38
TBK1 Q9UHD2 1/20 0.38
JAK1 P23458 1/20 0.38
MET P08581 3/20 0.37
HTR6 P50406 1/20 0.36
WNT1 P04628 1/20 0.36
GSK3B P49841 1/20 0.36
DYRK1A Q13627 1/20 0.36
CDK1 P06493 1/20 0.36
CDK4 P11802 1/20 0.36
CCNB1 P14635 1/20 0.36
CCND1 P24385 1/20 0.36
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25924724 0.91 MET (0.38) EGFRMAP3K7TAB1JAK1MET
SCHEMBL25924720 0.88 CYP1A2 (0.48) MAP3K7TAB1METMAP4K1
SCHEMBL25924718 0.85 TNK2 (0.49) EGFRMAP3K7TAB1METHTR6
SCHEMBL2283400 0.85 PDPK1 (0.42) HTR6WNT1GSK3BDYRK1ACDK2
SCHEMBL24723287 0.82 CYP3A4 (0.46) EGFRACVR1MAP3K7TAB1JAK1
SCHEMBL29273533 0.80 BMPR1A (0.42) EGFRACVR1BMPR1AACVRL1MAP3K7
SCHEMBL25926294 0.79 EGFR (0.37) EGFRMAP3K7TAB1MAP4K1
SCHEMBL24722970 0.79 JAK1 (0.39) EGFRACVR1BMPR1AACVRL1MAP3K7
SCHEMBL25925739 0.78 MET (0.37) EGFRMAP3K7TAB1JAK1MET
SCHEMBL25924810 0.77 MET (0.40) MAP3K7TAB1JAK1METHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131271-A1 PYRROLE FUSED-RING PYRAZOLE COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 杭州中美华东制药有限公司 2023-07-13 WO disclosed