SCHEMBL25926673

SCHEMBL25926673

Nc1ncc(O)c(CCc2ccccc2)n1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
ALDH1A1 P00352 2/20 0.51
HPGD P15428 2/20 0.51
MPO P05164 1/20 0.47
DAO P14920 1/20 0.45
MAPT P10636 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MAOA P21397 2/20 0.41
MAOB P27338 2/20 0.41
HSD17B10 Q99714 1/20 0.41
DHFR P00374 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7755586 0.80 MPO (0.47) KDM4EMPOMAOAMAOB
SCHEMBL6417219 0.77 DHFR (0.47) MAOAMAOBDHFR
SCHEMBL15400226 0.73 CYP2D6 (0.47) MAOBDHFR
SCHEMBL1317138 0.72 DHFR (0.54) DHFR
SCHEMBL30107620 0.72 DHFR (0.42) ALDH1A1MPODHFR
SCHEMBL10698612 0.70 MPO (0.47) MPO
SCHEMBL6415720 0.70 PIN1 (0.48) DHFR
SCHEMBL6379173 0.69 KDM4E (0.97) KDM4EALDH1A1HPGDMAPTHSD17B10
SCHEMBL6649038 0.69 HTR2C (0.48) KDM4EALDH1A1HPGDDAO
SCHEMBL27816217 0.69 APP (0.58) ALDH1A1HPGDMPOMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230242494-A1 MALONITRILE DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 2023-08-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242494-A1 MALONITRILE DERIVATIVES MAL2, ME1, C5 KDM4E 3238/4885ALDH1A1 20/4885HPGD 1793/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.