SCHEMBL25929683

SCHEMBL25929683

Cc1cc(Br)cnc1N1CCC(F)(F)CC1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 3/20 0.43
MBOAT4 Q96T53 1/20 0.36
OPRK1 P41145 9/20 0.35
PDE10A Q9Y233 1/20 0.34
CHRM3 P20309 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
WHR1 P49842 1/20 0.34
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
FLT3 P36888 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24215208 0.83 SCN10A (0.44) SCN10AMBOAT4OPRK1SIGMAR1PIK3CA
SCHEMBL30412557 0.81 TRPV1 (0.42) SCN10AMBOAT4PDE10ACHRM3PDE4A
SCHEMBL22803865 0.81 TRPV1 (0.42) SCN10AMBOAT4PDE10ACHRM3PDE4A
SCHEMBL2366907 0.79 HRH4 (0.48)
SCHEMBL30593370 0.79 HRH4 (0.48)
SCHEMBL1745337 0.78 KDM4E (0.36) OPRK1PIK3CAMTORFLT3
SCHEMBL15351824 0.78 SCN10A (0.36) SCN10APDE10ASIGMAR1PIK3CAMTOR
SCHEMBL24225614 0.78 ALDH1A3 (0.37) SCN10APDE10ASIGMAR1PIK3CAMTOR
SCHEMBL1707795 0.78 ALDH1A1 (0.44) OPRK1PDE10APIK3CAMTOR
SCHEMBL21905951 0.77 OPRK1 (0.57) SCN10AOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131271-A1 PYRROLE FUSED-RING PYRAZOLE COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 杭州中美华东制药有限公司 2023-07-13 WO disclosed