SCHEMBL2594641

SCHEMBL2594641

NC(=O)Cc1cn(Cc2ccc(C(F)(F)F)cc2)c2ccccc12

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ICMT O60725 14/20 0.65
HTR6 P50406 1/20 0.61
PLA2G2A P14555 2/20 0.57
ALDH1A1 P00352 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
GAA P10253 1/20 0.56
CYP2D6 P10635 1/20 0.56
MAPT P10636 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2595192 0.87 ICMT (0.74) ICMTPLA2G2AALDH1A1SMN1; SMN2
SCHEMBL8289938 0.86 PLA2G2A (0.74) ICMTPLA2G2AALDH1A1SMN1; SMN2
SCHEMBL4359581 0.84 HTR6 (0.69) HTR6ALDH1A1CYP1A2CYP3A4GAA
SCHEMBL8183003 0.83 ALDH1A1 (0.56) ICMTHTR6PLA2G2AALDH1A1CYP1A2
SCHEMBL3855663 0.82 HTR6 (0.57) ICMTHTR6ALDH1A1CYP1A2CYP3A4
SCHEMBL3855666 0.82 HTR6 (0.57) ICMTHTR6ALDH1A1CYP1A2CYP3A4
SCHEMBL8178374 0.81 HTR6 (0.62) ICMTHTR6ALDH1A1CYP1A2CYP3A4
SCHEMBL3850017 0.81 HTR6 (0.55) ICMTHTR6ALDH1A1CYP1A2CYP3A4
SCHEMBL4435107 0.81 PLA2G2A (0.57) ICMTHTR6PLA2G2AALDH1A1MAPT
SCHEMBL4927838 0.80 HTR6 (0.54) ICMTHTR6ALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011138265-A2 INDOLE AND INDAZOLE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS EVOTEC AG (DE) 2011-11-10 WO disclosed