SCHEMBL25958773

SCHEMBL25958773

CC1(O)CCN(C(=O)c2cc(N)c(C(=N)Br)cn2)CC1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.36
VNN1 O95497 1/20 0.36
TRPC6 Q9Y210 2/20 0.35
MTOR P42345 4/20 0.35
PIK3CA P42336 3/20 0.35
HIF1A Q16665 2/20 0.34
CYP3A4 P08684 2/20 0.34
USP2 O75604 1/20 0.34
CNR2 P34972 1/20 0.34
CYP2D6 P10635 1/20 0.34
HSD17B10 Q99714 2/20 0.33
GRM3 Q14832 1/20 0.33
CCR8 P51685 1/20 0.33
KCNH2 Q12809 1/20 0.33
F11 P03951 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
NAMPT P43490 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25958653 0.84 ALDH1A1 (0.42) CNR2ALDH1A1HPGDKMT2A
SCHEMBL25958758 0.81 ALOX5AP (0.38) TRPC6
SCHEMBL25958544 0.80 VNN1 (0.39) SCN9AVNN1TRPC6MTORPIK3CA
SCHEMBL25959270 0.79 SCN9A (0.40) SCN9AVNN1MTORPIK3CACYP3A4
SCHEMBL25958662 0.78 SMN1; SMN2 (0.45) VNN1HSD17B10ALDH1A1HPGD
SCHEMBL25958835 0.77 SCN9A (0.38) SCN9ATRPC6
SCHEMBL25958820 0.75 SMN1; SMN2 (0.36) HPGD
SCHEMBL25958792 0.72 VNN1 (0.40) VNN1HPGDKMT2A
SCHEMBL25958722 0.72 DPP4 (0.31) F11
SCHEMBL13388369 0.70 ALDH1A1 (0.46) SCN9AVNN1HIF1ACYP3A4USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3870582-B1 5-AZAINDAZOLE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 2023-07-19 EP disclosed