SCHEMBL25958820

SCHEMBL25958820

BC1(O)COCCN(C(=O)c2cc(N)c(C(=N)Br)cn2)C1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.36
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
ESR2 Q92731 1/20 0.33
GRM5 P41594 1/20 0.33
PDE4B Q07343 1/20 0.33
F10 P00742 1/20 0.31
LMNA P02545 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
NTRK1 P04629 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25958662 0.81 SMN1; SMN2 (0.45) SMN1; SMN2HPGDTSHRESR2GRM5
SCHEMBL25958792 0.77 VNN1 (0.40) SMN1; SMN2HPGDTSHRESR2GRM5
SCHEMBL25958653 0.75 ALDH1A1 (0.42) HPGDTSHRNPC1RAB9A
SCHEMBL25958773 0.75 SCN9A (0.36) HPGD
SCHEMBL25959308 0.73 LRRK2 (0.36) SMN1; SMN2HPGDTSHRESR2PDE4B
SCHEMBL25958568 0.73 SMN1; SMN2 (0.37) SMN1; SMN2HPGDTSHRESR2GRM5
SCHEMBL25958758 0.72 ALOX5AP (0.38)
SCHEMBL25958835 0.69 SCN9A (0.38)
SCHEMBL25958722 0.65 DPP4 (0.31)
SCHEMBL24058910 0.63 SMN1; SMN2 (0.36) SMN1; SMN2HPGDTSHRESR2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3870582-B1 5-AZAINDAZOLE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 2023-07-19 EP disclosed