SCHEMBL25968519

SCHEMBL25968519

CN(C)c1ccc(CNC2(C(=O)O)CC(C(=O)OC(C)(C)C)N(C(=O)OCC3c4ccccc4-c4ccccc43)C2)cc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.37
EPHX2 P34913 2/20 0.33
OPRD1 P41143 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 5/20 0.33
ALOX15 P16050 4/20 0.33
CYP3A4 P08684 3/20 0.33
KDM4E B2RXH2 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MAPT P10636 1/20 0.32
BACE1 P56817 1/20 0.32
FABP5 Q01469 2/20 0.32
FABP7 O15540 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
HSD17B10 Q99714 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP9 Q86TI2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25968518 0.94 CASP1 (0.39) CASP1EPHX2OPRD1BACE1FABP5
SCHEMBL25968525 0.91 CASP1 (0.37) CASP1EPHX2ALDH1A1BACE1FABP5
SCHEMBL25968601 0.90 CASP1 (0.37) CASP1EPHX2BACE1FABP5FABP7
SCHEMBL25344766 0.90 CASP1 (0.37) CASP1EPHX2BACE1FABP5FABP7
SCHEMBL25968589 0.89 NAMPT (0.37) CASP1EPHX2CYP3A4SMN1; SMN2TSHR
SCHEMBL25968522 0.88 SCN9A (0.43) CASP1
SCHEMBL25968596 0.88 CASP1 (0.36) CASP1EPHX2BACE1FABP5FABP7
SCHEMBL25343338 0.88 CASP1 (0.36) CASP1EPHX2BACE1FABP5FABP7
SCHEMBL25344636 0.88 CASP1 (0.36) CASP1EPHX2OPRD1SMN1; SMN2TSHR
SCHEMBL25968593 0.87 L3MBTL1 (0.35) CASP1L3MBTL1ALDH1A1CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154724-A2 PROCESSES AND COMPOUNDS FOR PREPARING SPIROLIGOMERS TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2023-08-17 WO disclosed