SCHEMBL2597597

SCHEMBL2597597

Clc1ncc(Oc2cccc(N3CCOCC3)c2)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.45
CNR2 P34972 4/20 0.45
AGXT P21549 1/20 0.45
LMNA P02545 1/20 0.44
KMO O15229 1/20 0.43
F10 P00742 1/20 0.43
AKR1C3 P42330 1/20 0.43
NTRK1 P04629 1/20 0.42
MAPT P10636 2/20 0.42
ALKBH1 Q13686 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
AKT1 P31749 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2597646 0.87 MAPT (0.42) DHFRAGXTLMNAF10MAPT
SCHEMBL2599593 0.86 AKR1C3 (0.45) DHFRCNR2AGXTLMNAKMO
SCHEMBL2599592 0.83 ADRA2C (0.49) DHFRAGXTMAPTALDH1A1
SCHEMBL3650599 0.83 F10 (0.44) DHFRCNR2AGXTLMNAKMO
SCHEMBL2599601 0.80 PIK3C3 (0.43) PIK3CAMTOR
SCHEMBL2599602 0.80 PIK3C3 (0.43) PIK3CAMTOR
SCHEMBL2599606 0.80 PIK3C3 (0.43) PIK3CAMTOR
SCHEMBL2597585 0.76 HDAC3 (0.48) NTRK1HDAC3HDAC1HDAC2HDAC6
SCHEMBL21345910 0.75 MAPK1 (0.50) AGXTLMNAKMOF10AKR1C3
SCHEMBL16621272 0.75 ALDH1A1 (0.56) DHFRAGXTLMNAKMOF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571872-B1 COMPOUNDS TREHERNE JOHNATHAN MARK (GB) 2014-12-31 EP disclosed
EP-2571872-B1 COMPOUNDS TREHERNE JOHNATHAN MARK (GB) 2014-12-31 EP disclosed
EP-2571872-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP disclosed
EP-2571856-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP disclosed
WO-2011144577-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed
WO-2011144578-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed