SCHEMBL2597946

SCHEMBL2597946

CC(C)COC(=O)C=P(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
TSHR P16473 3/20 0.49
HSP90AA1 P07900 1/20 0.46
HPGD P15428 2/20 0.41
P2RX4 Q99571 1/20 0.40
RAB9A P51151 1/20 0.38
LMNA P02545 2/20 0.38
CACNA1F O60840 1/20 0.37
CACNA1D Q01668 1/20 0.37
CACNA1S Q13698 1/20 0.37
CACNA1C Q13936 1/20 0.37
HSD17B10 Q99714 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 1/20 0.37
PLA2G1B P04054 1/20 0.37
ATG4B Q9Y4P1 1/20 0.37
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65066 0.81 HSP90AA1 (0.50) ALDH1A1TSHRHSP90AA1RAB9ALMNA
Bromide SCHEMBL6879691 0.80 HSP90AA1 (0.49) ALDH1A1TSHRHSP90AA1RAB9ALMNA
Hydrochloric Acid SCHEMBL9061399 0.80 HSP90AA1 (0.49) ALDH1A1TSHRHSP90AA1RAB9ALMNA
SCHEMBL2392064 0.79 LMNA (0.50) ALDH1A1TSHRHSP90AA1HPGDLMNA
SCHEMBL2392066 0.78 HSP90AA1 (0.46) ALDH1A1TSHRHSP90AA1RAB9ALMNA
SCHEMBL7907406 0.78 HSP90AA1 (0.54) ALDH1A1TSHRHSP90AA1LMNASMN1; SMN2
SCHEMBL2389657 0.77 HCAR2 (0.57) ALDH1A1TSHRHSP90AA1LMNASMN1; SMN2
SCHEMBL12305763 0.77 HCAR2 (0.57) ALDH1A1TSHRHSP90AA1LMNASMN1; SMN2
SCHEMBL852873 0.76 TSHR (0.50) ALDH1A1TSHRHSP90AA1HPGDLMNA
SCHEMBL9094 0.75 HSP90AA1 (0.50) ALDH1A1TSHRHSP90AA1HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571353-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF AbbVie Inc. (US) 2013-03-27 EP disclosed
WO-2011146089-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2011-11-24 WO disclosed