SCHEMBL2599340

SCHEMBL2599340

O=C1c2ccccc2C(=O)C(Cl)C1Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 3/20 1.00
KMT2A Q03164 7/20 0.55
MEN1 O00255 6/20 0.55
POLB P06746 2/20 0.55
MAPT P10636 5/20 0.50
LMNA P02545 2/20 0.50
TP53 P04637 2/20 0.50
MAPK1 P28482 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
HTR2B P41595 1/20 0.50
RAB9A P51151 4/20 0.48
PIM1 P11309 1/20 0.48
CDC25B P30305 1/20 0.45
IDO1 P14902 1/20 0.43
DNMT1 P26358 1/20 0.43
DNMT3L Q9UJW3 1/20 0.43
DNMT3A Q9Y6K1 1/20 0.43
NPC1 O15118 4/20 0.43
HTT P42858 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31237472 1.00 S100A4 (1.00) S100A4KMT2AMEN1POLBMAPT
SCHEMBL7645697 0.85 S100A4 (0.73) S100A4KMT2AMEN1POLBMAPT
SCHEMBL19147624 0.83 S100A4 (0.70) S100A4KMT2AMEN1POLBMAPT
SCHEMBL19130059 0.83 S100A4 (0.70) S100A4KMT2AMEN1POLBMAPT
SCHEMBL11595145 0.82 S100A4 (0.70) S100A4KMT2AMEN1POLBMAPT
SCHEMBL2126258 0.74 S100A4 (0.58) S100A4KMT2AMEN1POLBMAPT
SCHEMBL11741033 0.73 S100A4 (0.56) S100A4KMT2AMEN1POLBKDM4E
SCHEMBL9641853 0.72 S100A4 (0.56) S100A4RAB9APIM1CES1
SCHEMBL2205822 0.72 S100A4 (0.56) S100A4KMT2AMEN1POLBMAPT
SCHEMBL2599235 0.71 S100A4 (1.00) S100A4KMT2AMEN1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130090355-A1 CHEMICAL AGENTS FOR THE PREVENTION OF INHIBITION OR TUMOR METASTASIS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2013-04-11 US claimed
WO-2011146101-A1 CHEMICAL AGENTS FOR THE PREVENTION OR INHIBITION OF TUMOR METASTASIS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2011-11-24 WO claimed
JP-52151155-A None JP disclosed
US-20190022100-A1 ANTIVIRAL COMPOUNDS AND METHODS OF USE THEREOF TRANA DISCOVERY INC (US) 2019-01-24 US disclosed
CN-106831379-A A kind of method that 2,3 dichloro Isosorbide-5-Nitrae naphthoquinones are prepared with 2 chlorine Isosorbide-5-Nitrae naphthoquinones production process waste materials 天门楚天精细化工有限公司 2017-06-13 CN disclosed
US-20160129006-A1 ANTIVIRAL COMPOUNDS AND METHODS OF USE THEREOF TRANA DISCOVERY INC (US) 2016-05-12 US disclosed
US-20160129006-A1 ANTIVIRAL COMPOUNDS AND METHODS OF USE THEREOF TRANA DISCOVERY INC (US) 2016-05-12 US disclosed
US-9173886-B2 Antiviral compounds and methods of use thereof TRANA DISCOVERY, INC. (US) 2015-11-03 US disclosed
US-9173886-B2 Antiviral compounds and methods of use thereof TRANA DISCOVERY, INC. (US) 2015-11-03 US disclosed
US-20130090355-A1 CHEMICAL AGENTS FOR THE PREVENTION OF INHIBITION OR TUMOR METASTASIS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2013-04-11 US disclosed
US-20130090355-A1 CHEMICAL AGENTS FOR THE PREVENTION OF INHIBITION OR TUMOR METASTASIS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2013-04-11 US disclosed
WO-2010111718-A2 ANTIVIRAL COMPOUNDS AND METHODS OF USE THEREOF TRANA DISCOVERY (US) 2010-09-30 WO disclosed
WO-2005053609-A2 METHODS OF NAD+-DEPENDENT DEACETYLASE INHIBITORS GUILFORD PHARMACEUTICALS INC. (US) 2005-06-16 WO disclosed
EP-0062540-B1 PHOTOSENSITIVE COMPOSITION FOR ELECTROPHOTOGRAPHY MITA INDUSTRIAL CO. LTD. (JP) 1987-01-14 EP disclosed
EP-0088607-B1 ORGANIC PHOTOSENSITIVE MATERIAL FOR ELECTROPHOTOGRAPHY MITA INDUSTRIAL CO. LTD. (JP) 1986-07-16 EP disclosed
US-4447514-A PYRYLENE PIGMENT MITA INDUSTRIAL CO., LTD. (JP) 1984-05-08 US disclosed
US-4438187-A POLYVINYLCARBAZOLE, AND PERYLENE PIGMENT MITA INDUSTRIAL CO. LTD. (JP) 1984-03-20 US disclosed
EP-0088607-A2 Organic photosensitive material for electrophotography MITA INDUSTRIAL CO. LTD. (JP) 1983-09-14 EP disclosed
EP-0062540-A2 Photosensitive composition for electrophotography MITA INDUSTRIAL CO. LTD. (JP) 1982-10-13 EP disclosed
JP-S52151155-A PREPARATION OF 2,3-DIHYDRO-2,3-DICHLORO-1,4-NAPHTHOQUINONE KAWASAKI KASEI CHEM LTD 1977-12-15 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130090355-A1 CHEMICAL AGENTS FOR THE PREVENTION OF INHIBITION OR TUMOR METASTASIS S100A4, S100A6, S100A10 S100A4 1/4885KMT2A 3613/4885MEN1 1065/4885
US-20160129006-A1 ANTIVIRAL COMPOUNDS AND METHODS OF USE THEREOF TYMP, MAVS, ZC3HAV1 S100A4 4404/4885KMT2A 2800/4885MEN1 4495/4885
US-20190022100-A1 ANTIVIRAL COMPOUNDS AND METHODS OF USE THEREOF TYMP, MAVS, ZC3HAV1 S100A4 4404/4885KMT2A 2800/4885MEN1 4495/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.