SCHEMBL2599592

SCHEMBL2599592

CN1CCN(c2cccc(Oc3cnc(Cl)nc3)c2)CC1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.49
NPC1 O15118 2/20 0.46
MAPT P10636 2/20 0.46
AGXT P21549 1/20 0.45
EGFR P00533 1/20 0.45
HTR3A P46098 2/20 0.44
CTSC P53634 2/20 0.44
BRD4 O60885 1/20 0.43
KCNH2 Q12809 2/20 0.42
ALDH1A1 P00352 1/20 0.42
RAB9A P51151 1/20 0.42
MEN1 O00255 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
DHFR P00374 1/20 0.42
DRD2 P14416 1/20 0.42
HRH4 Q9H3N8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2597646 0.87 MAPT (0.42) NPC1MAPTAGXTHTR3AALDH1A1
SCHEMBL3656991 0.86 ADRA2C (0.47) ADRA2CNPC1MAPTAGXTEGFR
SCHEMBL2597597 0.83 DHFR (0.45) MAPTAGXTALDH1A1DHFR
SCHEMBL1040397 0.77 EGFR (0.56) ADRA2CNPC1MAPTEGFRCTSC
SCHEMBL28514042 0.75 SMN1; SMN2 (0.54) ADRA2CMAPTHTR3AALDH1A1MEN1
SCHEMBL28538439 0.75 HRH4 (0.45) HTR3AALDH1A1DRD2HRH4
SCHEMBL18938300 0.74 ADRA2C (0.59) ADRA2CNPC1MAPTAGXTHTR3A
SCHEMBL29814948 0.74 ADRA2C (0.59) ADRA2CNPC1MAPTAGXTHTR3A
SCHEMBL1372927 0.74 KCNH2 (0.69) ADRA2CNPC1MAPTAGXTHTR3A
SCHEMBL3653339 0.73 CHRNA3 (0.42) NPC1MAPTAGXTALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571872-B1 COMPOUNDS TREHERNE JOHNATHAN MARK (GB) 2014-12-31 EP disclosed
EP-2571872-B1 COMPOUNDS TREHERNE JOHNATHAN MARK (GB) 2014-12-31 EP disclosed
EP-2571872-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP disclosed
WO-2011144578-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed