SCHEMBL26027147

SCHEMBL26027147

O=c1[nH]nc(Oc2c(Cl)cc([N+](=O)[O-])cc2Cl)c2cc(Cl)c(Cl)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
HSD17B10 Q99714 1/20 0.37
RARG P13631 1/20 0.36
GRIN2D O15399 2/20 0.35
GRIN3B O60391 2/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2A Q12879 2/20 0.35
GRIN2B Q13224 2/20 0.35
GRIN2C Q14957 2/20 0.35
GRIN3A Q8TCU5 2/20 0.35
GPR35 Q9HC97 1/20 0.34
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
GALR3 O60755 1/20 0.33
PARP1 P09874 2/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
PDE7A Q13946 1/20 0.32
CA12 O43570 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29620356 0.87 RARG (0.46) ALDH1A1HSD17B10RARGPARP1MEN1
SCHEMBL26026549 0.87 RARG (0.46) ALDH1A1HSD17B10RARGPARP1MEN1
SCHEMBL26026709 0.82 RARG (0.46) ALDH1A1HSD17B10RARGGRIN2DGRIN3B
SCHEMBL29620364 0.82 ALDH1A1 (0.39) ALDH1A1HSD17B10GRIN2DGRIN3BGRIN1
SCHEMBL26027125 0.81 RARG (0.39) ALDH1A1HSD17B10RARGKMT2ATHRA
SCHEMBL27089947 0.79 PARP1 (0.45) ALDH1A1HSD17B10GPR35ADRA2AADRA2B
SCHEMBL26027642 0.77 TNKS (0.43) ALDH1A1RARGMEN1KMT2AMAPT
SCHEMBL29620357 0.76 ALDH1A1 (0.41) ALDH1A1HSD17B10GRIN2DGRIN3BGRIN1
SCHEMBL26027474 0.75 ALDH1A1 (0.33) ALDH1A1ADRA2AADRA2BADRA2C
SCHEMBL29620360 0.74 THRA (0.42) ALDH1A1MEN1KMT2ATHRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154842-A1 THR BETA ANALOGS AND USES THEREOF MADRIGAL PHARMACEUTICALS, INC. (US) 2023-08-17 WO disclosed