SCHEMBL260372

SCHEMBL260372

CCOC(=O)c1cccc2nc(N)sc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.51
HSD17B10 Q99714 5/20 0.51
TSHR P16473 1/20 0.50
RAB9A P51151 6/20 0.48
MAPT P10636 5/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
GAA P10253 3/20 0.48
HPGD P15428 3/20 0.48
ALOX15 P16050 2/20 0.48
CYP1A2 P05177 2/20 0.48
ILK Q13418 1/20 0.47
NPC1 O15118 5/20 0.45
KMT2A Q03164 4/20 0.45
MEN1 O00255 3/20 0.45
LMNA P02545 1/20 0.45
CDC25B P30305 3/20 0.45
MAPK1 P28482 1/20 0.43
TP53 P04637 1/20 0.43
CDC25A P30304 1/20 0.42
CDC25C P30307 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL261347 0.99 ALDH1A1 (0.50) ALDH1A1HSD17B10TSHRRAB9AMAPT
SCHEMBL19729156 0.89 ALDH1A1 (0.53) ALDH1A1HSD17B10TSHRRAB9AMAPT
SCHEMBL31053715 0.85 NPC1 (0.47) ALDH1A1RAB9AMAPTSMN1; SMN2HPGD
SCHEMBL1553043 0.84 TSHR (0.51) ALDH1A1HSD17B10TSHRRAB9AMAPT
SCHEMBL984327 0.84 ILK (0.59) ALDH1A1HSD17B10TSHRMAPTSMN1; SMN2
SCHEMBL6112936 0.83 TSHR (0.50) ALDH1A1HSD17B10TSHRRAB9AMAPT
SCHEMBL27998626 0.79 ASH1L (0.43) ALDH1A1HSD17B10RAB9AMAPTSMN1; SMN2
SCHEMBL9722823 0.78 ALDH1A1 (0.53) ALDH1A1HSD17B10TSHRRAB9AMAPT
SCHEMBL687318 0.77 ALDH1A1 (0.46) ALDH1A1HSD17B10RAB9AMAPTGAA
SCHEMBL2824199 0.77 PRKD3 (0.45) ALDH1A1HSD17B10TSHRRAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230159561-A1 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES FMC CORP (US) 2023-05-25 US disclosed
US-11578085-B2 Heterocycle-substituted bicyclic azole pesticides FMC CORPORATION (US) 2023-02-14 US disclosed
EP-4105209-A2 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES FMC Corporation (US) 2022-12-21 EP disclosed
EP-3424919-B1 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES FMC CORP (US) 2022-04-27 EP disclosed
CN-112679467-A Heterocyclic substituted bicyclic azoles as pesticidal agents FMC公司 2021-04-20 CN disclosed
CN-107635984-B Heterocyclic substituted bicyclic azoles as pesticidal agents FMC公司 2021-04-13 CN disclosed
CN-112608300-A Heterocyclic substituted bicyclic azoles as pesticidal agents FMC公司 2021-04-06 CN disclosed
US-20210017192-A1 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES FMC CORP (US) 2021-01-21 US disclosed
US-10822351-B2 Heterocycle-substituted bicyclic azole pesticides FMC CORPORATION (US) 2020-11-03 US disclosed
EP-3567036-A1 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES FMC Corporation (US) 2019-11-13 EP disclosed
US-20090209579-A1 INDAZOLES, BENZOTHIAZOLES, AND BENZOISOTHIAZOLES, AND PREPARATION AND USES THEREOF XIE WENGE 2009-08-20 US disclosed
US-7429664-B2 Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof MEMORY PHARMACEUTICALS CORPORATION (US) 2008-09-30 US disclosed
US-20080176890-A1 INDAZOLES, BENZOTHIAZOLES, AND BENZOISOTHIAZOLES, AND PREPARATION AND USES THEREOF XIE WENGE 2008-07-24 US disclosed
US-20080154037-A1 INDAZOLES, BENZOTHIAZOLES, AND BENZOISOTHIAZOLES, AND PREPARATION AND USES THEREOF XIE WENGE 2008-06-26 US disclosed
EP-1735306-A2 INDAZOLES, BENZOTHIAZOLES, BENZOISOTHIAZOLES, BENZISOXAZOLES, AND PREPARATION AND USES THEREOF Memory Pharmaceuticals Corporation (US) 2006-12-27 EP disclosed
US-20050234095-A1 Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof MEMORY PHARMACEUTICALS CORPORATION 2005-10-20 US disclosed
WO-2005092890-A2 INDAZOLES, BENZOTHIAZOLES, BENZOISOTHIAZOLES, BENZISOXAZOLES, AND PREPARATION AND USES THEREOF MEMORY PHARMACEUTICALS CORPORATION (US) 2005-10-06 WO disclosed
EP-1543000-A1 INDAZOLES, BENZOTHIAZOLES, AND BENZOISOTHIAZOLES, AND PREPARATION AND USES THEREOF Memory Pharmaceuticals Corporation (US) 2005-06-22 EP disclosed
US-20040132790-A1 Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof MEMORY PHARMACEUTICALS CORPORATION 2004-07-08 US disclosed
WO-2004029050-A1 INDAZOLES, BENZOTHIAZOLES, AND BENZOISOTHIAZOLES, AND PREPARATION AND USES THEREOF MEMORY PHARMACEUTICALS CORPORATION (US) 2004-04-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10822351-B2 Heterocycle-substituted bicyclic azole pesticides CYP4X1, DDT, CHRM1 ALDH1A1 2441/4885HSD17B10 2978/4885TSHR 1382/4885
US-20230159561-A1 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES CYP4X1, DDT, CHRM1 ALDH1A1 2441/4885HSD17B10 2978/4885TSHR 1382/4885
US-20040132790-A1 Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof CHRNA5, CHRNA7, CHRNA3 ALDH1A1 1431/4885HSD17B10 2432/4885TSHR 568/4885
US-11578085-B2 Heterocycle-substituted bicyclic azole pesticides CYP4X1, DDT, CHRM1 ALDH1A1 2441/4885HSD17B10 2978/4885TSHR 1382/4885
US-20090209579-A1 INDAZOLES, BENZOTHIAZOLES, AND BENZOISOTHIAZOLES, AND PREPARATION AND USES THEREOF CHRNA7, CHRNA5, CHRNA3 ALDH1A1 1268/4885HSD17B10 2300/4885TSHR 625/4885
US-20080154037-A1 INDAZOLES, BENZOTHIAZOLES, AND BENZOISOTHIAZOLES, AND PREPARATION AND USES THEREOF CHRNA7, CHRNA5, CHRNA3 ALDH1A1 1268/4885HSD17B10 2300/4885TSHR 625/4885
US-20080176890-A1 INDAZOLES, BENZOTHIAZOLES, AND BENZOISOTHIAZOLES, AND PREPARATION AND USES THEREOF CHRNA7, CHRNA5, CHRNA3 ALDH1A1 1268/4885HSD17B10 2300/4885TSHR 625/4885
US-20210017192-A1 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES CYP4X1, DDT, CHRM1 ALDH1A1 2441/4885HSD17B10 2978/4885TSHR 1382/4885
US-20050234095-A1 Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof CHRNA7, CHRNA5, CHRNA3 ALDH1A1 1806/4885HSD17B10 2288/4885TSHR 786/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.