SCHEMBL26058397

SCHEMBL26058397

COc1cccc(F)c1B1OC(C)(C)C(C)(C)O1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPL P06858 3/20 0.41
LIPG Q9Y5X9 3/20 0.41
NFE2L2 Q16236 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
BCHE P06276 2/20 0.36
ACHE P22303 2/20 0.36
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
KMT2A Q03164 1/20 0.34
EGFR P00533 2/20 0.34
HPGD P15428 2/20 0.33
RPS6KA2 Q15349 1/20 0.33
NPC1 O15118 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22505969 0.89 LPL (0.38) LPLLIPGJAK2BTK
SCHEMBL28915005 0.88 CA1 (0.41) LPLLIPGTDP1CA12CA1
SCHEMBL15026275 0.84 LPL (0.46) LPLLIPGCA12CA1CA2
SCHEMBL22972610 0.83 LPL (0.36) LPLLIPGL3MBTL1TDP1JAK2
SCHEMBL30191147 0.83 L3MBTL1 (0.44) LPLLIPGL3MBTL1TDP1KMT2A
SCHEMBL21296144 0.83 LPL (0.38) LPLLIPGKMT2AJAK2BTK
SCHEMBL29574505 0.83 LPL (0.38) LPLLIPGKMT2AJAK2BTK
SCHEMBL22534910 0.81 LPL (0.37) LPLLIPGJAK2BTK
SCHEMBL26647695 0.81 CSF1R (0.38) LPLLIPGACHECA12CA1
SCHEMBL24558106 0.81 AR (0.37) LPLLIPGNFE2L2L3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12410183-B2 Sars-cov2 main protease inhibitors GILEAD SCIENCES, INC. (US) 2025-09-09 US disclosed
US-20250042915-A1 SARS-COV2 MAIN PROTEASE INHIBITORS GILEAD SCIENCES, INC. 2025-02-06 US disclosed
US-20250026766-A1 Thiazolopyridyl Amide Derivatives as DNA Polymerase Theta Inhibitors BEIGENE, LTD. (KY) 2025-01-23 US disclosed
EP-4463456-A1 THIAZOLOPYRIDYL AMIDE DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS BeiGene, Ltd. (KY) 2024-11-20 EP disclosed
US-12091420-B2 SARS-COV2 main protease inhibitors GILEAD SCIENCES, INC. (US) 2024-09-17 US disclosed
US-20240239807-A1 SARS-COV2 MAIN PROTEASE INHIBITORS GILEAD SCIENCES, INC. 2024-07-18 US disclosed
US-20240116946-A1 SARS-COV2 MAIN PROTEASE INHIBITORS GILEAD SCIENCES, INC. 2024-04-11 US disclosed
US-11731958-B2 Carboxamide compounds and uses thereof INCYTE CORPORATION (US) 2023-08-22 US disclosed
WO-2023134708-A1 THIAZOLOPYRIDYL AMIDE DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS BEIGENE , LTD. (KY) 2023-07-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250042915-A1 SARS-COV2 MAIN PROTEASE INHIBITORS ACE2, TMPRSS2, ACE LPL 230/4885LIPG 232/4885NFE2L2 859/4885
US-12091420-B2 SARS-COV2 main protease inhibitors ACE2, TMPRSS2, ACE LPL 230/4885LIPG 232/4885NFE2L2 859/4885
US-20240116946-A1 SARS-COV2 MAIN PROTEASE INHIBITORS ACE2, TMPRSS2, ACE LPL 230/4885LIPG 232/4885NFE2L2 859/4885
US-12410183-B2 Sars-cov2 main protease inhibitors ACE2, TMPRSS2, ACE LPL 230/4885LIPG 232/4885NFE2L2 859/4885
US-11731958-B2 Carboxamide compounds and uses thereof PCK1, PHKG2, PHKG1 LPL 2908/4885LIPG 3259/4885NFE2L2 1369/4885
US-20240239807-A1 SARS-COV2 MAIN PROTEASE INHIBITORS ACE2, TMPRSS2, ACE LPL 230/4885LIPG 232/4885NFE2L2 859/4885
US-20250026766-A1 Thiazolopyridyl Amide Derivatives as DNA Polymerase Theta Inhibitors POLQ, POLK, POLI LPL 2850/4885LIPG 2760/4885NFE2L2 2535/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.