SCHEMBL26075166

SCHEMBL26075166

CCCNS(=O)(=O)c1c(F)cc(F)c(F)c1F

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.44
CA2 P00918 5/20 0.44
CA9 Q16790 4/20 0.44
CA12 O43570 3/20 0.41
CA7 P43166 1/20 0.37
CA13 Q8N1Q1 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
POLB P06746 1/20 0.35
PNMT P11086 2/20 0.34
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26501949 0.86 CA1 (0.42) CA1CA2CA9CA12CA7
SCHEMBL26075086 0.82 CA1 (0.43) CA1CA2CA9CA12L3MBTL1
SCHEMBL15453138 0.77 CA1 (0.49) CA1CA2CA9CA12CA7
SCHEMBL26075094 0.76 CA1 (0.39) CA1CA2CA9CA12CA7
SCHEMBL26075093 0.75 PKM (0.50) CA1CA2CA9CA12POLB
SCHEMBL26075285 0.74 CA1 (0.51) CA1CA2CA9CA12CA7
SCHEMBL25359552 0.70 CA2 (0.38) CA1CA2CA9CA12
SCHEMBL3687291 0.69 L3MBTL1 (0.61) CA1CA2L3MBTL1POLB
SCHEMBL6186899 0.68 CYP3A4 (0.54) CA1CA2CA9CA12L3MBTL1
SCHEMBL3528445 0.67 CA12 (0.58) CA9CA12L3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11976075-B2 Inhibitors of the MYST family of lysine acetyl transferases Isosterix, Inc. 2024-05-07 US disclosed
US-20230303580-A1 INHIBITORS OF THE MYST FAMILY OF LYSINE ACETYL TRANSFERASES Isosterix, Inc. 2023-09-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303580-A1 INHIBITORS OF THE MYST FAMILY OF LYSINE ACETYL TRANSFERASES KAT6A, KAT6B, KAT2A CA1 3845/4885CA2 4141/4885CA9 3963/4885
US-11976075-B2 Inhibitors of the MYST family of lysine acetyl transferases KAT6A, KAT6B, KAT2A CA1 3845/4885CA2 4141/4885CA9 3963/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.