SCHEMBL26093046

SCHEMBL26093046

NC(=O)Oc1ccc(CO)nc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
MEN1 O00255 1/20 0.41
KIF11 P52732 1/20 0.38
PARP10 Q53GL7 5/20 0.35
PARP15 Q460N3 1/20 0.35
MAPT P10636 1/20 0.34
PIK3CA P42336 1/20 0.33
PI4KA P42356 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
FFAR1 O14842 1/20 0.32
P4HTM Q9NXG6 1/20 0.32
KCNH2 Q12809 1/20 0.32
ATM Q13315 1/20 0.32
GRM2 Q14416 1/20 0.32
NNMT P40261 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
CCR1 P32246 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28292626 0.86 KMT2A (0.39) KMT2AMEN1KIF11PARP10MAPT
SCHEMBL28375297 0.86 KMT2A (0.41) KMT2AMEN1KIF11PARP10PARP15
SCHEMBL29273373 0.84 MEN1 (0.54) KMT2AMEN1PARP10PARP15
SCHEMBL9519545 0.81 AOC3 (0.39) KMT2AMEN1KIF11PARP10MAPT
SCHEMBL2904971 0.81 POLB (0.44) KMT2AMEN1MAPT
SCHEMBL26640548 0.79 SYK (0.39) KMT2AMEN1KIF11PARP10MAPT
SCHEMBL28292573 0.79 KIF11 (0.36) KMT2AMEN1KIF11PARP10MAPT
SCHEMBL5568443 0.78 RAB9A (0.56) KMT2AMEN1SMN1; SMN2
SCHEMBL28286228 0.78 KMT2A (0.49) KMT2AMEN1KIF11PARP10PARP15
SCHEMBL27691370 0.77 NNMT (0.53) KMT2AMEN1KIF11NNMTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116554092-A Method for preparing new drug building block (6-formylpyridin-3-yl) carbamic acid tert-butyl ester 上海锐谱医药科技有限公司 2023-08-08 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-118119626-A Fused bicyclic heteroaryl compounds useful as NLRP3 inhibitors 豪夫迈·罗氏有限公司 2024-05-31 CN disclosed
CN-116554092-A Method for preparing new drug building block (6-formylpyridin-3-yl) carbamic acid tert-butyl ester 上海锐谱医药科技有限公司 2023-08-08 CN disclosed
CN-116554092-A Method for preparing new drug building block (6-formylpyridin-3-yl) carbamic acid tert-butyl ester 上海锐谱医药科技有限公司 2023-08-08 CN disclosed
WO-2023066825-A1 FUSED BICYCLIC HETEROARYL COMPOUNDS USEFUL AS NLRP3 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2023-04-27 WO disclosed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-110770224-B Indole derivatives as efflux pump inhibitors 罗格斯新泽西州立大学 2022-11-18 CN disclosed
CN-110770224-A Indole derivatives as efflux pump inhibitors 罗格斯新泽西州立大学 2020-02-07 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed
CN-104394869-A Substituted bicyclic aza-heterocycles and analogues as sirtuin modulators GLAXOSMITHKLINE LLC 2015-03-04 CN disclosed