SCHEMBL8934162

SCHEMBL8934162

COC(=O)c1nccnc1N.COC(=O)c1nccnc1N(CCCl)C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.39
TDP1 Q9NUW8 1/20 0.39
KDM4E B2RXH2 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
GBA1 P04062 1/20 0.34
RCE1 Q9Y256 1/20 0.34
PRKCI P41743 3/20 0.33
PIK3CD O00329 1/20 0.33
ATR Q13535 1/20 0.33
GRM4 Q14833 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8708337 0.94 L3MBTL1 (0.36) NPC1TDP1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL32682741 0.78 NPSR1 (0.48) NPC1TDP1KDM4ERAB9ASMN1; SMN2
SCHEMBL261104 0.78 NPSR1 (0.48) NPC1TDP1KDM4ERAB9ASMN1; SMN2
SCHEMBL7857665 0.77 KDM4E (0.33) KDM4EALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL5773639 0.76 NPSR1 (0.46) NPC1TDP1KDM4ERAB9ASMN1; SMN2
SCHEMBL71518 0.65 NPSR1 (0.59) TDP1KDM4ESMN1; SMN2ALDH1A1GAA
SCHEMBL29133980 0.65 L3MBTL1 (0.41) KDM4ESMN1; SMN2ALDH1A1GAAL3MBTL1
SCHEMBL13482134 0.64 TMPRSS15 (0.41) RAB9ASMN1; SMN2ALDH1A1L3MBTL1GBA1
SCHEMBL29642902 0.64 RAB9A (0.55) NPC1TDP1KDM4ERAB9ASMN1; SMN2
SCHEMBL3979132 0.64 RAB9A (0.55) NPC1TDP1KDM4ERAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022991-A1 BICYCLIC SUBSTITUTED HEXAHYDROBENZ[E]ISOINDOLE ALPHA-1- ADRENERGIC ANTAGONISTS ABBOTT LABORATORIES (US) 1996-08-01 WO disclosed