Fluproquazone

Fluproquazone

SCHEMBL26210

Cc1ccc2c(-c3ccc(F)cc3)nc(=O)n(C(C)C)c2c1

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.77
EGFR P00533 1/20 0.77
ADRA2A P08913 1/20 0.77
ADORA3 P0DMS8 1/20 0.77
TBXA2R P21731 1/20 0.77
PTGS2 P35354 1/20 0.77
OPRD1 P41143 1/20 0.77
PDE4D Q08499 1/20 0.77
CASR P41180 18/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluproquazone SCHEMBL29363976 1.00 NR1I2 (0.77) NR1I2EGFRADRA2AADORA3TBXA2R
SCHEMBL11565990 0.92 NR1I2 (0.85) NR1I2EGFRADRA2AADORA3TBXA2R
SCHEMBL11723933 0.87 NR1I2 (0.77) NR1I2EGFRADRA2AADORA3TBXA2R
Proquazone SCHEMBL29508590 0.87 NR1I2 (1.00) NR1I2EGFRADRA2AADORA3TBXA2R
Proquazone SCHEMBL25341 0.87 NR1I2 (1.00) NR1I2EGFRADRA2AADORA3TBXA2R
Proquazone SCHEMBL2931942 0.86 NR1I2 (0.97) NR1I2EGFRADRA2AADORA3TBXA2R
Fluproquazone SCHEMBL11080399 0.84 NR1I2 (0.61) NR1I2EGFRADRA2AADORA3TBXA2R
SCHEMBL11726950 0.83 NR1I2 (0.54) NR1I2EGFRADRA2AADORA3TBXA2R
SCHEMBL11608840 0.81 NR1I2 (0.67) NR1I2EGFRADRA2AADORA3TBXA2R
SCHEMBL11605525 0.79 NR1I2 (0.76) NR1I2EGFRADRA2AADORA3TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1912 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260000741-A1 METHOD OF AMELIORATING A PRO-INFLAMMATORY IMMUNOPHENOTYPE IN FARBER DISEASE SUBJECTS BY REPEATED ADMINISTRATION OF A RECOMBINANT HUMAN ACID CERAMIDASE ACERAGEN INC (US) 2026-01-01 US claimed
EP-3998932-A1 ALKALIZATION OF URINARY BLADDER WALL PRIOR TO TREATMENT WITH INTRAVESICAL HEPARIN AND ALKALINIZED LIDOCAINE TO ENHANCE RELIEF OF BLADDER PAIN SYMPTOMS Parsons, C. Lowell (US) 2022-05-25 EP claimed
US-20220088158-A1 METHOD OF AMELIORATING A PRO-INFLAMMATORY IMMUNOPHENOTYPE IN FARBER DISEASE SUBJECTS BY REPEATED ADMINISTRATION OF A RECOMBINANT HUMAN ACID CERAMIDASE ROIVANT SCIENCES, INC. 2022-03-24 US claimed
WO-2021011566-A1 ALKALIZATION OF URINARY BLADDER WALL PRIOR TO TREATMENT WITH INTRAVESICAL HEPARIN AND ALKALINIZED LIDOCAINE TO ENHANCE RELIEF OF BLADDER PAIN SYMPTOMS PARSONS C LOWELL (US) 2021-01-21 WO claimed
WO-2020152532-A1 METHOD OF AMELIORATING A PRO-INFLAMMATORY IMMUNOPHENOTYPE IN FARBER DISEASE SUBJECTS BY REPEATED ADMINISTRATION OF A RECOMBINANT HUMAN ACID CERAMIDASE ENZYVANT THERAPEUTICS GMBH (CH) 2020-07-30 WO claimed
EP-3609483-A1 ARTICLE OF MANUFACTURE COMPRISING LOCAL ANESTHETIC, BUFFER, AND GLYCOSAMINOGLYCAN IN SYRINGE WITH IMPROVED STABILITY Urigen Pharmaceuticals, Inc. (US) 2020-02-19 EP claimed
WO-2018191412-A9 ARTICLE OF MANUFACTURE COMPRISING LOCAL ANESTHETIC, BUFFER, AND GLYCOSAMINOGLYCAN IN SYRINGE WITH IMPROVED STABILITY URIGEN PHARMACEUTICALS, INC. (US) 2019-05-31 WO claimed
WO-2018191412-A1 ARTICLE OF MANUFACTURE COMPRISING LOCAL ANESTHETIC, BUFFER, AND GLYCOSAMINOGLYCAN IN SYRINGE WITH IMPROVED STABILITY URIGEN PHARMACEUTICALS, INC. (US) 2018-10-18 WO claimed
EP-3351262-A1 CURAGLUTIDE FOR IN TREATMENT OF PREDIABETES, DIABETES, OBESITY AND METABOLIC DISEASES ASSOCIATED THERETO Istanbul Universitesi Rektorlugu (TR) 2018-07-25 EP claimed
US-20160113936-A1 METHODS FOR MODULATING MONOCYTE FUNCTION AUGUSTA UNIVERSITY RESEARCH INSTITUTE, INC. 2016-04-28 US claimed
WO-2004082719-A1 DISPERSIBLE PHARMACEUTICAL COMPOSITION FOR TREATMENT OF MASTITIS AND OTIC DISORDERS PHARMACIA CORPORATION (US) 2004-09-30 WO claimed
US-20040156872-A1 Novel nimesulide compositions ELAN PHARMA INTERNATIONAL LTD. 2004-08-12 US claimed
US-20030235617-A1 Pharmaceutical dosage form for mucosal delivery MCNEIL-PPC, INC 2003-12-25 US claimed
US-20030180357-A1 Pharmaceutical tablet MCNEIL-PPC, INC 2003-09-25 US claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
WO-2003066029-A2 PHARMACEUTICAL DOSAGE FORM FOR MUCOSAL DELIVERY PHARMACIA CORPORATION (US) 2003-08-14 WO claimed
WO-2003066030-A2 PHARMACEUTICAL TABLET PHARMACIA CORPORATION (US) 2003-08-14 WO claimed
US-4442084-A ABSORPTION, LIQUID PHASE CLAUS PROCESS, RECYCLING SANDOZ LTD. (CH) 1984-04-10 US claimed
US-4236006-A Preparation of quinazolin-2(1H)-ones SANDOZ LTD. (CH) 1980-11-25 US claimed
US-4224328-A Methods with 1-substituted-4-aryl-quinazolin-2(1H)-ones and thiones and pyrido[2,3-d]pyrimidin-2-ones as platelet aggregation inhibitors SANDOZ, INC. (US) 1980-09-23 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040156872-A1 Novel nimesulide compositions NIM1K, NIT2, NCL NR1I2 3919/4885EGFR 2788/4885ADRA2A 3740/4885
US-20030180357-A1 Pharmaceutical tablet GYPA, SORD, SRI NR1I2 1613/4885EGFR 4459/4885ADRA2A 1648/4885
US-20030235617-A1 Pharmaceutical dosage form for mucosal delivery SI, UGGT1, GYPA NR1I2 1375/4885EGFR 2803/4885ADRA2A 1503/4885
US-20160113936-A1 METHODS FOR MODULATING MONOCYTE FUNCTION CD14, HSP90AB2P, HSP90AB1 NR1I2 967/4885EGFR 4841/4885ADRA2A 2670/4885
US-20260000741-A1 METHOD OF AMELIORATING A PRO-INFLAMMATORY IMMUNOPHENOTYPE IN FARBER DISEASE SUBJECTS BY REPEATED ADMINISTRATION OF A RECOMBINANT HUMAN ACID CERAMIDASE ASAH2, ASAH1, GBA2 NR1I2 1617/4885EGFR 4492/4885ADRA2A 2411/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.