SCHEMBL26212980

SCHEMBL26212980

O=S(=O)(NCCCl)c1ccc(-c2c(F)cccc2F)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT6A Q92794 1/20 0.47
NEK1 Q96PY6 3/20 0.46
PKM P14618 5/20 0.45
ALDH1A1 P00352 4/20 0.45
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
TAAR1 Q96RJ0 1/20 0.43
KDM4E B2RXH2 2/20 0.43
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 1/20 0.43
CYP3A4 P08684 1/20 0.41
PKLR P30613 3/20 0.41
CYP19A1 P11511 1/20 0.41
TDO2 P48775 1/20 0.41
GAA P10253 1/20 0.40
MMP2 P08253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26212993 0.90 NEK1 (0.49) KAT6ANEK1PKMALDH1A1KMT2A
SCHEMBL30270495 0.88 KIF11 (0.41) KAT6ANEK1PKMALDH1A1KMT2A
SCHEMBL26213011 0.88 KIF11 (0.41) KAT6ANEK1PKMALDH1A1KMT2A
SCHEMBL26217944 0.87 NEK1 (0.51) KAT6ANEK1PKMALDH1A1KMT2A
SCHEMBL26212996 0.84 GRIA4 (0.56) KAT6APKMALDH1A1KMT2AMEN1
SCHEMBL26212913 0.79 MMP2 (0.60) KAT6APKMALDH1A1TAAR1KDM4E
SCHEMBL20522284 0.79 ALDH1A1 (0.70) PKMALDH1A1KMT2AMEN1TAAR1
SCHEMBL26217870 0.78 NEK1 (0.55) NEK1PKMALDH1A1KMT2AKDM4E
SCHEMBL24196028 0.76 CA12 (0.49) KAT6APKMALDH1A1KMT2AMEN1
SCHEMBL26213025 0.76 PKM (0.40) KAT6ANEK1PKMALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12570632-B2 Indole derivatives and uses thereof for treating a cancer UNIVERSITE CLAUDE BERNARD LYON 1 (FR) 2026-03-10 US disclosed
EP-4175718-B1 INDOLE DERIVATIVES AND USES THEREOF FOR TREATING A CANCER UNIV CLAUDE BERNARD LYON (FR) 2024-10-02 EP disclosed
CN-115843271-B Indole derivatives and their use for the treatment of cancer 克洛德贝纳尔-里昂第一大学 2024-08-13 CN disclosed
US-20230278983-A1 INDOLE DERIVATIVES AND USES THEREOF FOR TREATING A CANCER UNIVERSITE CLAUDE BERNARD LYON 1 (FR) 2023-09-07 US disclosed
US-20230278983-A1 INDOLE DERIVATIVES AND USES THEREOF FOR TREATING A CANCER UNIVERSITE CLAUDE BERNARD LYON 1 (FR) 2023-09-07 US disclosed
US-20230278983-A1 INDOLE DERIVATIVES AND USES THEREOF FOR TREATING A CANCER UNIVERSITE CLAUDE BERNARD LYON 1 (FR) 2023-09-07 US disclosed
EP-4175718-A1 INDOLE DERIVATIVES AND USES THEREOF FOR TREATING A CANCER UNIVERSITE CLAUDE BERNARD - LYON 1 (FR) 2023-05-10 EP disclosed
CN-115843271-A Indole derivatives and their use for the treatment of cancer 克洛德贝纳尔-里昂第一大学 2023-03-24 CN disclosed
WO-2022008475-A1 INDOLE DERIVATIVES AND USES THEREOF FOR TREATING A CANCER UNIVERSITE CLAUDE BERNARD LYON 1 (FR) 2022-01-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12570632-B2 Indole derivatives and uses thereof for treating a cancer CKS2, CSNK2A3, CSNK1A1L KAT6A 199/4885NEK1 912/4885PKM 1790/4885
US-20230278983-A1 INDOLE DERIVATIVES AND USES THEREOF FOR TREATING A CANCER CSNK2A1, IDO1, CSNK2A3 KAT6A 882/4885NEK1 288/4885PKM 502/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.