SCHEMBL26219682

SCHEMBL26219682

CCCCCn1ccc(-c2ccc(N=O)cc2)n1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.44
TLR8 Q9NR97 10/20 0.36
KEAP1 Q14145 1/20 0.35
MGAT2 Q10469 1/20 0.35
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24168945 0.81 KEAP1 (0.57) CYP19A1TLR8KEAP1KMT2A
SCHEMBL6431328 0.80 KMT2A (0.55) CYP19A1TLR8KMT2A
SCHEMBL26215154 0.78 LMNA (0.45) CYP19A1KMT2A
SCHEMBL11679229 0.76 CYP19A1 (0.49) CYP19A1TLR8KEAP1KMT2A
SCHEMBL28782368 0.76 KEAP1 (0.59) CYP19A1TLR8KEAP1KMT2A
SCHEMBL29933067 0.75 CYP19A1 (0.39) CYP19A1TLR8MGAT2
SCHEMBL28903876 0.74 CYP19A1 (0.47) CYP19A1TLR8KEAP1KMT2A
SCHEMBL27753624 0.74 CYP19A1 (0.47) CYP19A1TLR8KEAP1KMT2A
SCHEMBL27753622 0.73 APOBEC3G (0.49) CYP19A1KMT2A
SCHEMBL24168406 0.72 THRA (0.52) CYP19A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230286904-A1 INHIBITORS OF YAP/TAZ-TEAD ONCOPROTEINS, SYNTHESIS AND USE THEREOF BRIDGENE BIOSCIENCES, INC. 2023-09-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230286904-A1 INHIBITORS OF YAP/TAZ-TEAD ONCOPROTEINS, SYNTHESIS AND USE THEREOF TEAD1, TEAD2, TEAD3 CYP19A1 4193/4885TLR8 4806/4885KEAP1 65/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.