SCHEMBL2625323

SCHEMBL2625323

[2H]c1ccc(-c2nc(C)c3c(n2)CCN(CCC)C3=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.39
DRD2 P14416 3/20 0.39
HTR2A P28223 3/20 0.39
PKN2 Q16513 1/20 0.34
GRM5 P41594 2/20 0.33
ADK P55263 1/20 0.32
LMNA P02545 1/20 0.31
PARP1 P09874 1/20 0.31
HTT P42858 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
ALDH1A1 P00352 2/20 0.30
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30
TLR9 Q9NR96 1/20 0.30
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
ALOX15 P16050 1/20 0.30
RAB9A P51151 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10220350 0.87 HTR1A (0.39) HTR1ADRD2HTR2APKN2GRM5
SCHEMBL13423652 0.84 GRM5 (0.36) HTR1ADRD2HTR2AGRM5ADK
SCHEMBL2625330 0.68 TLR9 (0.40) PKN2LMNAALDH1A1ADORA3ADORA2A
SCHEMBL2625325 0.67 HSF1 (0.35) HTR2AADKLMNAHTTALDH1A1
SCHEMBL2625327 0.62 KCNH2 (0.36) LMNAALDH1A1ADORA3ADORA2AADORA1
SCHEMBL13423651 0.61 TDP2 (0.39) HTR2AADKLMNAHTTALDH1A1
SCHEMBL2625321 0.60 DRD2 (0.43) DRD2LMNATLR9KCNH2
SCHEMBL2625322 0.60 TDP2 (0.40) LMNAALDH1A1ADORA3ADORA2AADORA1
SCHEMBL2625305 0.60 ALDH1A1 (0.40) HTR2AALDH1A1ADORA3ADORA2AADORA1
SCHEMBL4747714 0.60 MAPK1 (0.39) GRM5HTTALDH1A1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163763-B2 Pyrimidine compounds, compositions and methods of use GENENTECH, INC. (US) 2012-04-24 US disclosed