Aminopyrine

Aminopyrine

SCHEMBL26293

Cc1c(N(C)C)c(=O)n(-c2ccccc2)n1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 3/20 1.00
LMNA P02545 2/20 1.00
CYP1A2 P05177 1/20 1.00
THRB P10828 1/20 1.00
TSHR P16473 1/20 1.00
NAPRT Q6XQN6 1/20 1.00
PTGS1 P23219 1/20 0.63
MAPT P10636 2/20 0.62
KDM4E B2RXH2 1/20 0.62
ALOX12 P18054 1/20 0.62
HSD17B10 Q99714 2/20 0.61
BCHE P06276 8/20 0.60
ALDH1A1 P00352 2/20 0.60
PTGS2 P35354 1/20 0.60
POLB P06746 1/20 0.59
ADORA3 P0DMS8 1/20 0.58
GAA P10253 1/20 0.56
MEN1 O00255 1/20 0.55
PSMD14 O00487 1/20 0.55
NPC1 O15118 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Aminopyrine SCHEMBL1331641 1.00 ALOX15 (1.00) ALOX15LMNACYP1A2THRBTSHR
Aminopyrine SCHEMBL10489978 1.00 ALOX15 (1.00) ALOX15LMNACYP1A2THRBTSHR
Aminopyrine SCHEMBL2818734 0.98 ALOX15 (0.97) ALOX15LMNACYP1A2THRBTSHR
Aminopyrine SCHEMBL8723416 0.92 ALOX15 (0.85) ALOX15LMNACYP1A2THRBTSHR
Aminopyrine SCHEMBL28152267 0.92 ALOX15 (0.85) ALOX15LMNACYP1A2THRBTSHR
Aminopyrine SCHEMBL10493337 0.90 ALOX15 (0.81) ALOX15LMNACYP1A2THRBTSHR
Propyphenazone SCHEMBL28086369 0.90 LMNA (0.81) ALOX15LMNACYP1A2THRBTSHR
Aminopyrine SCHEMBL28086243 0.89 ALOX15 (0.78) ALOX15LMNACYP1A2THRBTSHR
Aminopyrine SCHEMBL7042293 0.84 ALOX15 (0.71) ALOX15LMNACYP1A2THRBTSHR
SCHEMBL13243351 0.84 ALOX15 (0.72) ALOX15LMNACYP1A2THRBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 9091 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260130928-A1 COMBINATION OF AKR1C3 ACTIVATED ANTICANCER PRODRUG COMPOUND AND ANALGESIC DRUG FOR TREATING CANCER PATIENTS ACCOMPANIED BY PAIN ASCENTAWITS PHARMACEUTICALS LTD (CN) 2026-05-14 US claimed
US-20260083666-A1 METHOD OF TREATING DISEASE CREWS THOMAS M (US) 2026-03-26 US claimed
US-20260069532-A1 METHOD FOR MORSELIZING AND/OR TARGETING PHARMACEUTICALLY ACTIVE PRINCIPLES TO SYNOVIAL TISSUE MEDINCELL S.A. (FR) 2026-03-12 US claimed
US-12558309-B2 Method for morselizing and/or targeting pharmaceutically active principles to synovial tissue MEDINCELL S.A. (FR) 2026-02-24 US claimed
US-20260000741-A1 METHOD OF AMELIORATING A PRO-INFLAMMATORY IMMUNOPHENOTYPE IN FARBER DISEASE SUBJECTS BY REPEATED ADMINISTRATION OF A RECOMBINANT HUMAN ACID CERAMIDASE ACERAGEN INC (US) 2026-01-01 US claimed
EP-3480730-B1 3D ANISOTROPIC HYBRID NETWORK: TRANSFERRING CONVOLUTIONAL FEATURES FROM 2D IMAGES TO 3D ANISOTROPIC VOLUMES Siemens Healthineers Ag (DE) 2025-11-26 EP claimed
WO-2025224317-A1 A METHOD FOR TARGETING PHARMACEUTICALLY ACTIVE PRINCIPLE IN TOTAL KNEE REPLACEMENT MEDINCELL S.A. (FR) 2025-10-30 WO claimed
EP-4630574-A1 TEST SYSTEM FOR MEASURING THE ENZYME ACTIVITY OF ANGIOTENSIN-CONVERTING ENZYME (ACE) DiaSys Diagnostic Systems GmbH (DE) 2025-10-15 EP claimed
EP-4182532-B1 FURNITURE FITTING FOR MOUNTING A FURNITURE PART BLUM GMBH JULIUS (AT) 2025-09-24 EP claimed
US-20250255781-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-08-14 US claimed
EP-0311616-A4 COMBINATIONS OF GAMMA INTERFERONS AND ANTI-INFLAMMATORY OR ANTI-PYRETIC AGENTS FOR TREATING DISEASES. BIOGEN NV (NL) 1989-05-23 EP claimed
EP-0311616-A1 COMBINATIONS OF GAMMA INTERFERONS AND ANTI-INFLAMMATORY OR ANTI-PYRETIC AGENTS FOR TREATING DISEASES. BIOGEN NV (NL) 1989-04-19 EP claimed
US-4757016-A Adding aminopyrine as stabilizer BOEHRINGER MANNHEIM GMBH (DE) 1988-07-12 US claimed
WO-1987007842-A1 COMBINATIONS OF GAMMA INTERFERONS AND ANTI-INFLAMMATORY OR ANTI-PYRETIC AGENTS AND METHODS FOR TREATING DISEASES BIOGEN N.V. (AN) 1987-12-30 WO claimed
EP-0147780-A2 Drug delivery device MERCK & CO. INC. (US) 1985-07-10 EP claimed
EP-0036145-B1 AN ORALLY ADMINISTERED DRUG FORM COMPRISING A POLAR BIOACTIVE AGENT AND AN ADJUVANT INTERx RESEARCH CORPORATION (US) 1985-05-29 EP claimed
EP-0129893-A2 Ground mixture Takeda Chemical Industries, Ltd. (JP) 1985-01-02 EP claimed
US-4420476-A Benzofuro[3,2-c]pyrazol-3-amine derivatives Averst McKenna & Harrison, Inc. (CA) 1983-12-13 US claimed
US-4350762-A BLOCKING INTERFERENCE BY BILITRUBIN ELVI S.P.A. (IT) 1982-09-21 US claimed
EP-0033462-A1 Aminopyrine improved Trinder's reagent and dosing process for hydrogen peroxide from enzimatic oxidation of metabolic substrata with the same ELVI S.p.A. (IT) 1981-08-12 EP claimed