SCHEMBL263096

SCHEMBL263096

Brc1cccc2c1OCO2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.50
AOC3 Q16853 1/20 0.44
HTR2A P28223 2/20 0.43
HTR2C P28335 1/20 0.43
GSK3B P49841 1/20 0.40
PKM P14618 1/20 0.39
TSHR P16473 1/20 0.39
EED O75530 1/20 0.38
TTBK1 Q5TCY1 1/20 0.36
TTBK2 Q6IQ55 1/20 0.36
TXNRD1 Q16881 1/20 0.35
TXNRD3 Q86VQ6 1/20 0.35
TXNRD2 Q9NNW7 1/20 0.35
MAOB P27338 2/20 0.35
POLB P06746 2/20 0.35
MAPK1 P28482 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29523159 1.00 ABCG2 (0.50) ABCG2AOC3HTR2AHTR2CGSK3B
SCHEMBL31452716 0.83 ABCG2 (0.41) ABCG2AOC3HTR2AHTR2CPKM
SCHEMBL4564550 0.82 ITGB2 (0.50) MAPK1KDM4EALDH1A1LMNAHTR1A
SCHEMBL38654029 0.78 ITGB2 (0.41) MAOBKDM4EALDH1A1LMNA
SCHEMBL31454272 0.78 ABCG2 (0.31) ABCG2HTR2AHTR2CHTR1A
SCHEMBL30583926 0.78 ABCG2 (0.31) ABCG2HTR2AHTR2CHTR1A
SCHEMBL7594061 0.76 ABCG2 (0.55) ABCG2GSK3BPKMTSHREED
SCHEMBL30521296 0.74 ABCG2 (0.52) ABCG2GSK3BPKMTSHREED
SCHEMBL1224045 0.74 ABCG2 (0.52) ABCG2GSK3BPKMTSHREED
SCHEMBL2168952 0.74 EED (0.46) ABCG2AOC3HTR2AHTR2CGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 180 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106749204-A A kind of preparation method of piribedil 郑州大明药物科技有限公司 2017-05-31 CN claimed
US-20080249128-A1 Substituted Sulfonamide Compounds GRUENENTHAL GMBH (DE) 2008-10-09 US claimed
CN-122036680-A Anti-fibrotic pyridones 英特穆恩公司 2026-05-15 CN disclosed
EP-4317162-B1 1,3-BENZODIOXOLANE-CONTAINING COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF XIAN XINTONG PHARMACEUTICAL RES CO LTD (CN) 2026-02-04 EP disclosed
US-20260022096-A1 NOVEL SULFONAMIDES AND THEIR USE AS NEUROPROTECTIVE AND/OR NEURORESTORATIVE AGENTS GENECODE (EE) 2026-01-22 US disclosed
US-12435060-B2 Acylamino bridged heterocyclic compound, and composition and application thereof BEIJING SCITECH-MQ PHARMACEUTICALS LIMITED (CN) 2025-10-07 US disclosed
US-20250296915-A1 NOVEL AMINO ACID DERIVATIVES PEPTIDREAM INC (JP) 2025-09-25 US disclosed
US-20250179046-A1 SEROTONIN 5-HT2B INHIBITORY COMPOUNDS ZOETIS SERVICES LLC 2025-06-05 US disclosed
EP-4561994-A1 NOVEL SULFONAMIDES AND THEIR USE AS NEUROPROTECTIVE AND/OR NEURORESTORATIVE AGENTS Genecode (EE) 2025-06-04 EP disclosed
US-12240827-B2 Serotonin 5-HT2B inhibitory compounds ZOETIS SERVICES LLC (US) 2025-03-04 US disclosed
US-20250026766-A1 Thiazolopyridyl Amide Derivatives as DNA Polymerase Theta Inhibitors BEIGENE, LTD. (KY) 2025-01-23 US disclosed
US-4978801-A Preparation of aromatic aldehydes RHONE-POULENC CHIMIE (FR) 1990-12-18 US disclosed
US-4942240-A REACTION OF HYDROGEN AND CARBON MONOXIDE WITH AN AROMATIC HALIDE IN THE PRESENCE OF A NOBLE METAL CATALYSTS RHONE-POULENC CHIMIE (FR) 1990-07-17 US disclosed
US-4746358-A PLANT GROWTH REGULATORS, HERBICIDES; N-TRIAZINYL-AMINOCARBONYL -1,4-BENZODIOXANESULFONAMIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 1988-05-24 US disclosed
EP-0244328-A2 Process for the preparation of aromatic aldehydes RHONE-POULENC CHIMIE (FR) 1987-11-04 EP disclosed
EP-0244329-A2 Process for the preparation of aromatic aldehydes RHONE-POULENC CHIMIE (FR) 1987-11-04 EP disclosed
US-4659368-A HERBICIDES; PLANT GROWTH REGULATORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-04-21 US disclosed
US-4595407-A Triazinyl-amino-carbonyl-1,3-benzohetero- or -1,4-benzohetero-sulfonamides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1986-06-17 US disclosed
US-4502882-A HERBICIDES, PLANT GROWTH REGULATORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1985-03-05 US disclosed
EP-0082681-A2 Herbicidal sulfonamides E.I. DU PONT DE NEMOURS AND COMPANY (US) 1983-06-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12240827-B2 Serotonin 5-HT2B inhibitory compounds HTR2B, HTR1B, HTR5A ABCG2 273/4885AOC3 2550/4885HTR2A 9/4885
US-20250179046-A1 SEROTONIN 5-HT2B INHIBITORY COMPOUNDS HTR2B, HTR1B, HTR5A ABCG2 273/4885AOC3 2550/4885HTR2A 9/4885
US-20250296915-A1 NOVEL AMINO ACID DERIVATIVES DNPEP, BCAT1, ANPEP ABCG2 842/4885AOC3 4644/4885HTR2A 3126/4885
US-20260022096-A1 NOVEL SULFONAMIDES AND THEIR USE AS NEUROPROTECTIVE AND/OR NEURORESTORATIVE AGENTS CNR1, CDR2, SMN1; SMN2 ABCG2 684/4885AOC3 768/4885HTR2A 1496/4885
US-20080249128-A1 Substituted Sulfonamide Compounds BDKRB1, BDKRB2, NPSR1 ABCG2 350/4885AOC3 3678/4885HTR2A 464/4885
US-20250026766-A1 Thiazolopyridyl Amide Derivatives as DNA Polymerase Theta Inhibitors POLQ, POLK, POLI ABCG2 3423/4885AOC3 3492/4885HTR2A 4540/4885
US-12435060-B2 Acylamino bridged heterocyclic compound, and composition and application thereof RIPK1, RIPK3, RIPK4 ABCG2 1665/4885AOC3 4463/4885HTR2A 4631/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.