SCHEMBL263115

SCHEMBL263115

FC(F)(F)Cc1ccccc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.46
IDO1 P14902 2/20 0.45
TSHR P16473 2/20 0.38
NR3C1 P04150 1/20 0.38
CYP2A13 Q16696 1/20 0.37
PYCR1 P32322 1/20 0.36
RIPK1 Q13546 1/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA5A P35218 1/20 0.35
CA9 Q16790 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
NFKB1 P19838 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SLC6A2 P23975 1/20 0.35
LMNA P02545 1/20 0.34
BLM P54132 1/20 0.34
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11717665 0.82 IDO1 (0.38) TAAR1IDO1TSHRRIPK1ALDH1A1
SCHEMBL11066668 0.77 TAAR1 (0.54) TAAR1IDO1TSHRCYP2A13PYCR1
SCHEMBL7847384 0.76 TRPA1 (0.35) IDO1TSHRALDH1A1
SCHEMBL1691374 0.76 RIPK1 (0.47) TAAR1IDO1TSHRNR3C1CYP2A13
SCHEMBL5697510 0.73 TAAR1 (0.43) TAAR1IDO1TSHRCYP2A13PYCR1
SCHEMBL15638695 0.73 TAAR1 (0.50) TAAR1IDO1TSHRNR3C1CYP2A13
SCHEMBL18623577 0.73 TAAR1 (0.44) TAAR1IDO1TSHRNR3C1CYP2A13
SCHEMBL2401345 0.73 RIPK1 (0.45) TAAR1IDO1TSHRNR3C1CYP2A13
SCHEMBL30388724 0.73 RIPK1 (0.45) TAAR1IDO1TSHRNR3C1CYP2A13
SCHEMBL28754249 0.73 TAAR1 (0.44) TAAR1IDO1TSHRNR3C1CYP2A13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 56 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260085073-A1 PYRAZOLYLCARBOXAMIDE COMPOUNDS AND THEIR USE IN THERAPY HOTSPOT THERAPEUTICS INC (US) 2026-03-26 US disclosed
EP-4540238-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME Monte Rosa Therapeutics AG (CH) 2025-04-23 EP disclosed
US-20250115582-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME MONTE ROSA THERAPEUTICS AG (CH) 2025-04-10 US disclosed
US-20240101553-A1 KRAS G12C INHIBITORS MIRATI THERAPEUTICS INC (US) 2024-03-28 US disclosed
WO-2024059524-A1 PYRAZOLYLCARBOXAMIDE COMPOUNDS AND THEIR USE IN THERAPY HOTSPOT THERAPEUTICS, INC. (US) 2024-03-21 WO disclosed
WO-2023244818-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME MONTE ROSA THERAPEUTICS, INC. (US) 2023-12-21 WO disclosed
US-20230373999-A1 KRAS G12C INHIBITORS MIRATI THERAPEUTICS INC (US) 2023-11-23 US disclosed
EP-3710439-B1 KRAS G12C INHIBITORS MIRATI THERAPEUTICS INC (US) 2023-02-15 EP disclosed
US-11267812-B2 KRAS G12C inhibitors Mirati Therapeutics, Inc. (US) 2022-03-08 US disclosed
CN-112500517-A Oil-soluble super-heavy oil viscosity reducer and preparation method and application thereof 山东德仕化工有限公司 2021-03-16 CN disclosed
CN-101516884-A Octahydropyrrolo [3, 4-C] pyrrole derivatives an their use as antiviral agents HOFFMANN LA ROCHE (CH) 2009-08-26 CN disclosed
US-20090048306-A1 PYRIDINE DERIVATIVES PFIZER, INC. (US) 2009-02-19 US disclosed
US-20090048306-A1 PYRIDINE DERIVATIVES PFIZER, INC. (US) 2009-02-19 US disclosed
US-20090048306-A1 PYRIDINE DERIVATIVES PFIZER, INC. (US) 2009-02-19 US disclosed
WO-2008135826-A2 2 -PYRIDINE CARBOXAMIDE DERIVATIVES AS SODIUM CHANNEL MODULATORS PFIZER LIMITED (GB) 2008-11-13 WO disclosed
WO-2008135826-A2 2 -PYRIDINE CARBOXAMIDE DERIVATIVES AS SODIUM CHANNEL MODULATORS PFIZER LIMITED (GB) 2008-11-13 WO disclosed
CN-101084198-A Substituted amino-pyrimidones and uses thereof ASTRAZENECA AB (SE) 2007-12-05 CN disclosed
CN-101084199-A Substituted amino-compounds and uses thereof ASTRAZENECA AB (SE) 2007-12-05 CN disclosed
CN-101039947-A Inhibitors of hcv replication BRISTOL MYERS SQUIBB CO (US) 2007-09-19 CN disclosed
CN-1894235-A N-(4-carbamimidoyl-benzyl) -2-alkoxy-2-heterocyclyl acetamides as inhibitors of the formation of coagulation factors xa, ixa and thrombin induced by factor viia HOFFMANN LA ROCHE (CH) 2007-01-10 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11267812-B2 KRAS G12C inhibitors KRAS, NRAS, HRAS TAAR1 4854/4885IDO1 4640/4885TSHR 4273/4885
US-20240101553-A1 KRAS G12C INHIBITORS KRAS, NRAS, HRAS TAAR1 4854/4885IDO1 4640/4885TSHR 4273/4885
US-20090048306-A1 PYRIDINE DERIVATIVES SDHA, P2RX4, P2RX3 TAAR1 1946/4885IDO1 1538/4885TSHR 3678/4885
US-20260085073-A1 PYRAZOLYLCARBOXAMIDE COMPOUNDS AND THEIR USE IN THERAPY MALT1, BCL6, BCL3 TAAR1 3408/4885IDO1 392/4885TSHR 2143/4885
US-20250115582-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME PSMA1, CSNK1G1, CSNK1A1 TAAR1 2209/4885IDO1 3139/4885TSHR 4501/4885
US-20230373999-A1 KRAS G12C INHIBITORS KRAS, NRAS, HRAS TAAR1 4854/4885IDO1 4640/4885TSHR 4273/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.