Metazocine

Metazocine

SCHEMBL26347

CC1C2Cc3ccc(O)cc3C1(C)CCN2C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 8/20 1.00
OPRD1 P41143 7/20 1.00
OPRK1 P41145 7/20 1.00
SIGMAR1 Q99720 7/20 1.00
MRGPRX2 Q96LB1 2/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Metazocine SCHEMBL13353229 1.00 OPRM1 (1.00) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
Metazocine SCHEMBL21994208 1.00 OPRM1 (1.00) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
Metazocine SCHEMBL12013732 1.00 OPRM1 (1.00) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
Metazocine SCHEMBL1649365 1.00 OPRM1 (1.00) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
Metazocine SCHEMBL12049577 1.00 OPRM1 (1.00) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
Metazocine SCHEMBL29387774 1.00 OPRM1 (1.00) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL15866689 0.92 SIGMAR1 (0.85) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL12267534 0.84 SIGMAR1 (0.73) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL12324824 0.84 SIGMAR1 (0.73) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL12716235 0.84 SIGMAR1 (0.73) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 7111 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4724049-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF Catalent Ontario Limited (CA) 2026-04-15 EP claimed
US-12564597-B2 Ibogaine analogs as therapeutics for neurological and psychiatric disorders THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE OF NEW YORK (US) 2026-03-03 US claimed
US-20250319074-A1 TREATMENT AND MANAGEMENT OF AUGMENTATION IN RESTLESS LEGS SYNDROME UNIV EAST CAROLINA (US) 2025-10-16 US claimed
US-12383743-B2 Treatment of addiction and dependency TACA JR ARTURO C (US) 2025-08-12 US claimed
US-20250228771-A1 ALKALINE INTRAORAL PRODUCTS EMPLICURE AB (publ) (SE) 2025-07-17 US claimed
EP-4581017-A1 NEW N-HETEROARYLBENZAMIDES DERIVATIVES AS FLT3 INHIBITORS Biodol Therapeutics (FR) 2025-07-09 EP claimed
EP-4565202-A1 ALKALINE INTRAORAL PRODUCTS EMPLICURE AB (publ) (SE) 2025-06-11 EP claimed
WO-2024254056-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF CATALENT ONTARIO LIMITED (CA) 2024-12-12 WO claimed
US-12133922-B2 Abuse resistant capsule R.P. SCHERER TECHNOLOGIES, LLC (US) 2024-11-05 US claimed
CN-118647367-A Novel injectable combination formulations 南爱克萨股份公司 2024-09-13 CN claimed
US-4882335-A Method for treating alcohol-drinking response ALKO LIMITED (FI) 1989-11-21 US claimed
EP-0046270-B1 NOVEL DERIVATIVES OF BIO-AFFECTING PHENOLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM INTERx RESEARCH CORPORATION (US) 1986-05-21 EP claimed
US-4546103-A Method of treating weight loss disorders HUEBNER HANS F 1985-10-08 US claimed
US-4464378-A Method of administering narcotic antagonists and analgesics and novel dosage forms containing same UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 1984-08-07 US claimed
US-4434168-A Narcotic antagonists in the therapy of shock THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 1984-02-28 US claimed
EP-0077393-A1 NOVEL METHOD OF ADMINISTERING NARCOTIC ANTAGONISTS AND ANALGESICS AND NOVEL DOSAGE FORMS CONTAINING SAME The University of Kentucky Research Foundation (US) 1983-04-27 EP claimed
WO-1982003768-A1 NOVEL METHOD OF ADMINISTERING NARCOTIC ANTAGONISTS AND ANALGESICS AND NOVEL DOSAGE FORMS CONTAINING SAME UNIV KENTUCKY (US) 1982-11-11 WO claimed
EP-0046270-A1 Novel derivatives of bio-affecting phenolic compounds and pharmaceutical composition containing them INTERx RESEARCH CORPORATION (US) 1982-02-24 EP claimed
US-4267182-A Narcotic antagonists in the therapy of shock THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 1981-05-12 US claimed
US-4126684-A 4-AMINO-3-P-HALOPHENYLBUTYRIC ACIDS AND THEIR DERIVATIVES USED IN THE CONTROL OF NARCOTIC ABUSE CIBA-GEIGY CORPORATION (US) 1978-11-21 US claimed