SCHEMBL2637580

SCHEMBL2637580

O=C(Nc1c(=O)[nH]n2c(=O)cc(-c3ccccc3)[nH]c12)c1ccccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.44
HDAC1 Q13547 1/20 0.42
NOX4 Q9NPH5 1/20 0.42
NOX1 Q9Y5S8 1/20 0.42
KDM4E B2RXH2 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
LMNA P02545 1/20 0.40
ALDH1A1 P00352 1/20 0.39
ADRB2 P07550 1/20 0.39
PKM P14618 1/20 0.39
KDR P35968 2/20 0.39
KCNK3 O14649 1/20 0.39
KCNK9 Q9NPC2 1/20 0.39
ERCC1 P07992 1/20 0.38
FEN1 P39748 1/20 0.38
ERCC4 Q92889 1/20 0.38
GRM4 Q14833 2/20 0.38
HDAC6 Q9UBN7 1/20 0.38
ADORA2A P29274 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2637343 0.85 ALDH1A1 (0.46) GRM5MEN1KMT2AALDH1A1ERCC1
SCHEMBL2637556 0.80 POLB (0.46) KDM4EMEN1KMT2ALMNAALDH1A1
SCHEMBL2637547 0.80 NPC1 (0.48) GRM5MEN1KMT2ALMNAPKM
SCHEMBL2637908 0.80 NPC1 (0.45) GRM5HDAC1NOX4NOX1KDM4E
SCHEMBL2637478 0.79 HSP90AA1 (0.47) GRM5MEN1KMT2ALMNAALDH1A1
SCHEMBL2637595 0.75 MAPT (0.43) GRM5MEN1KMT2ALMNAPKM
SCHEMBL2637716 0.74 KMT2A (0.47) KDM4EMEN1KMT2ALMNAALDH1A1
SCHEMBL2638043 0.74 MAPK10 (0.45) MEN1KMT2AKDRERCC1FEN1
SCHEMBL2638375 0.74 MAPT (0.48) GRM5MEN1KMT2ALMNAALDH1A1
SCHEMBL2637610 0.73 MAPK8 (0.48) KDM4EMEN1KMT2ALMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2438070-A1 GLYCINE B ANTAGONISTS Merz Pharma GmbH & Co. KGaA (DE) 2012-04-11 EP disclosed
WO-2010139483-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2010-12-09 WO disclosed