SCHEMBL2637556

SCHEMBL2637556

O=C(Nc1c(=O)[nH]n2c(=O)cc(-c3ccc(Cl)cc3)[nH]c12)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
PSD A5PKW4 3/20 0.46
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C19 P33261 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MAPT P10636 2/20 0.44
HSP90AA1 P07900 1/20 0.44
HSP90AB1 P08238 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
SUCNR1 Q9BXA5 1/20 0.40
MET P08581 1/20 0.39
KDR P35968 1/20 0.39
MEN1 O00255 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2637343 0.92 ALDH1A1 (0.46) POLBTDP1ALDH1A1SMN1; SMN2NPC1
SCHEMBL2637478 0.89 HSP90AA1 (0.47) POLBTDP1PSDALDH1A1NPC1
SCHEMBL2637595 0.85 MAPT (0.43) TDP1SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL2637889 0.83 KMT2A (0.46) POLBALDH1A1KDM4ENPC1RAB9A
SCHEMBL2637590 0.82 KDM4E (0.41) ALDH1A1KDM4ECYP1A2CYP2C19SMN1; SMN2
SCHEMBL2637740 0.80 KDM5A (0.41) TDP1ALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL2637580 0.80 GRM5 (0.44) TDP1ALDH1A1KDM4EKDRMEN1
SCHEMBL2637547 0.78 NPC1 (0.48) POLBTDP1SMN1; SMN2NPC1RAB9A
SCHEMBL2637406 0.77 MAPT (0.41) TDP1ALDH1A1KDM4ESMN1; SMN2NPC1
SCHEMBL2638047 0.77 KDM4A (0.44) POLBPSDALDH1A1KDM4ECYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2438070-A1 GLYCINE B ANTAGONISTS Merz Pharma GmbH & Co. KGaA (DE) 2012-04-11 EP disclosed
WO-2010139483-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2010-12-09 WO disclosed