SCHEMBL264299

SCHEMBL264299

FC(F)Oc1ccccc1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 1/20 0.42
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
KMT2A Q03164 2/20 0.41
HTT P42858 2/20 0.41
MEN1 O00255 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.39
HTR7 P34969 1/20 0.38
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
SLC22A12 Q96S37 1/20 0.35
POLB P06746 1/20 0.35
ALOX12 P18054 1/20 0.35
NR1I2 O75469 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
KDM4E B2RXH2 1/20 0.34
PTGES2 Q9H7Z7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29819809 1.00 DRD1 (0.42) DRD1HTR1AADRA2AADRA2BADRA2C
SCHEMBL22823665 0.82 HTR1A (0.46) HTR1AADRA2AADRA2BADRA2CKMT2A
SCHEMBL1400223 0.82 HTR1A (0.39) HTR1AADRA2AADRA2BADRA2CKMT2A
SCHEMBL4654255 0.82 DRD1 (0.48) DRD1KMT2AHTTSMN1; SMN2ALDH1A1
SCHEMBL29867899 0.80 HTT (0.41) DRD1KMT2AHTTMEN1SMN1; SMN2
SCHEMBL28310793 0.80 IDO1 (0.39) HTR1AADRA2AADRA2BADRA2CKMT2A
SCHEMBL2031163 0.80 HTT (0.41) DRD1KMT2AHTTMEN1SMN1; SMN2
SCHEMBL25435045 0.79 ALDH1A1 (0.42) DRD1KMT2AHTTMEN1SMN1; SMN2
SCHEMBL8984707 0.79 HTR1A (0.37) HTR1AADRA2AADRA2BADRA2CKMT2A
SCHEMBL31399767 0.79 KMT2A (0.40) DRD1KMT2AHTTMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 130 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106083602-A A kind of synthetic method of phenformin pharmaceutical intermediate β phenethylamine 成都切斯特科技有限公司 2016-11-09 CN claimed
US-12630566-B2 KRas G12D inhibitors Mirati Therapeutics, Inc. (US) 2026-05-19 US disclosed
US-20260109715-A1 IMIDAZOPYRIDINE DERIVATIVES WITH BICYCLIC STRUCTURE PUBLIC UNIVERSITY CORPORATION YOKOHAMA CITY UNIVERSITY (JP) 2026-04-23 US disclosed
US-20260055062-A1 HETEROCYCLIC INHIBITORS OF MCT4 Vettore, LLC 2026-02-26 US disclosed
US-20260049074-A1 THIADIAZOLYL DERIVATIVES IDEAYA BIOSCIENCES, INC. (US) 2026-02-19 US disclosed
US-12509454-B2 Thiadiazolyl derivatives IDEAYA BIOSCIENCES, INC. (US) 2025-12-30 US disclosed
US-12492171-B2 Heterocyclic inhibitors of MCT4 Vettore, LLC (US) 2025-12-09 US disclosed
US-20250325552-A1 SUBSTITUTED THIADIAZOLYL DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS IDEAYA BIOSCIENCES INC (US) 2025-10-23 US disclosed
EP-4600246-A1 IMIDAZOPYRIDINE DERIVATIVES WITH BICYCLIC STRUCTURE Public University Corporation Yokohama City University (JP) 2025-08-13 EP disclosed
EP-4587014-A2 C5AR1 ANTAGONISTS AND USES THEREOF Vanqua Bio, Inc. (US) 2025-07-23 EP disclosed
WO-2003018535-A2 NOVEL AMINOBENZOEPHENONES LEO PHARMA A/S (DK) 2003-03-06 WO disclosed
EP-0393513-B1 Preparation of a difluorohalomethoxybenzene MITSUI TOATSU CHEMICALS (JP) 1994-03-09 EP disclosed
US-5105021-A Reacting metal phenolate with (di)bromo(chloro)difluoromethane in presence of promoter MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1992-04-14 US disclosed
EP-0393513-A1 Preparation of a difluorohalomethoxybenzene MITSUI TOATSU CHEMICALS, Inc. (JP) 1990-10-24 EP disclosed
EP-0147298-B1 SULFONYLATION PROCESS RHONE-POULENC CHIMIE (FR) 1989-04-26 EP disclosed
US-4618726-A DEACTIVATED BENZENE COMPOUND WITH CARBONYL HALIDE IN LIQUID HYDROFLUORIC ACID AND BORON TRIFLUORIDE RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1986-10-21 US disclosed
EP-0147298-A2 Sulfonylation process RHONE-POULENC CHIMIE (FR) 1985-07-03 EP disclosed
EP-0052558-B1 AROMATIC BROMOPOLYFLUOROALKYL ETHERS, AND PROCESS FOR THEIR PREPARATION RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1984-10-03 EP disclosed
US-4377711-A Novel aromatic bromopolyfluoroalkyl ethers and method for the preparation thereof RHONE-POULENC INDUSTRIES (FR) 1983-03-22 US disclosed
EP-0052558-A1 Aromatic bromopolyfluoroalkyl ethers, and process for their preparation RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1982-05-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12492171-B2 Heterocyclic inhibitors of MCT4 SLC16A3, SLC16A1, MCTS1 DRD1 4758/4885HTR1A 2313/4885ADRA2A 4616/4885
US-20260049074-A1 THIADIAZOLYL DERIVATIVES POLH, POLM, POLD1 DRD1 2052/4885HTR1A 2674/4885ADRA2A 838/4885
US-20250325552-A1 SUBSTITUTED THIADIAZOLYL DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS POLQ, POLK, POLH DRD1 4199/4885HTR1A 4304/4885ADRA2A 3026/4885
US-12630566-B2 KRas G12D inhibitors KRAS, NRAS, HRAS DRD1 3863/4885HTR1A 4856/4885ADRA2A 4569/4885
US-20260109715-A1 IMIDAZOPYRIDINE DERIVATIVES WITH BICYCLIC STRUCTURE SMG1, RACK1, TIA1 DRD1 2544/4885HTR1A 3198/4885ADRA2A 3086/4885
US-12509454-B2 Thiadiazolyl derivatives POLD1, POLQ, DNA2 DRD1 769/4885HTR1A 2705/4885ADRA2A 1621/4885
US-20260055062-A1 HETEROCYCLIC INHIBITORS OF MCT4 SLC16A1, SLC16A3, SLC16A7 DRD1 1700/4885HTR1A 627/4885ADRA2A 3965/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.